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N-(2-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)acetamide
N-[(5-{[2-(methylsulfanyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
3-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
8-(2-fluorobenzoyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
2-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]acetamide
2-(1-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1H-imidazol-2-yl)-1-methyl-1H-imidazole
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-5-hydroxy-1,2-dimethyl-1H-indole-3-carboxamide
1-[3-({[(2-methoxynaphthalen-1-yl)methyl]amino}methyl)pyridin-2-yl]piperidin-3-ol
(1S,5R)-6-(1H-indole-6-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-4-(2-phenoxyethyl)piperazine
3-{[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}piperidine
(2-{[(6-methoxypyridin-3-yl)methyl][(2-methylphenyl)methyl]amino}ethyl)dimethylamine
3-(1-{[1-(6-chloropyridazin-3-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-1-ol
3-[(4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1H-1,2,3-triazol-1-yl)methyl]piperidine
(4aS,7aR)-1-(3-phenylpropanoyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-({[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}(thiophen-3-ylmethyl)amino)butan-1-ol
(1S,3R)-3-amino-N-{2-[2-(trifluoromethoxy)phenyl]ethyl}cyclopentane-1-carboxamide
2-methoxy-5-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]pyrimidine
dimethyl({[(1R,5S,6S)-3-{[2-(prop-2-yn-1-yloxy)phenyl]methyl}-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
1-(2-methoxyphenyl)-3-{[1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]methyl}urea
5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
(3aS,6aS)-2-[(3,4-dichlorophenyl)methyl]-5-(2-methoxyacetyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-({2-[1-(3-chloro-5-fluorobenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
3-(2,4-dimethoxybenzoyl)-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidine
8-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-(4-chlorophenyl)-2-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(3R,4R)-1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
(4R)-N,3-dimethyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,3-thiazolidine-4-carboxamide
4-{4-[3-(3-ethylphenoxy)azetidin-1-yl]piperidin-1-yl}-6-methylpyrimidin-2-amine
1-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}propan-2-yl)piperidine
4-(methoxymethyl)-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)benzamide
N-[(4-fluorophenyl)methyl]-1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
N-[(2-tert-butyl-6-oxo-1,6-dihydropyrimidin-4-yl)methyl]-N'-(2,5-dimethylphenyl)ethanediamide
6-{[2-(2-oxoimidazolidin-1-yl)ethyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-hydroxy-2-methylpropan-2-yl)acetamide
5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-2,1,3-benzoxadiazole
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
N-[(4,6-dimethylpyridin-3-yl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
(2S,4R)-1-{2-[4-(dimethylamino)phenyl]acetyl}-N-ethyl-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
3-(3-ethyl-3-hydroxypiperidin-1-yl)-N-(4-methoxy-2-methylphenyl)propanamide
methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)[(2E)-2-methylbut-2-en-1-yl]amine
5-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]-2-(pyridin-2-yl)pyrimidin-4-ol
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-(1-methyl-1H-pyrazol-4-yl)propanamide
4-[(4-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}-1H-1,2,3-triazol-1-yl)methyl]-N-(2-methylphenyl)piperidine-1-carboxamide
3-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-fluorophenyl)urea
1-(2-{[2-(3-methylthiophen-2-yl)ethyl]amino}pyrimidin-4-yl)pyrrolidin-3-ol
4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-N-(2-phenylethyl)pyrimidin-2-amine
(3R,4R)-1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
7-fluoro-3-[1-(6-methylpyridin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one