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1-[(1R,5R)-6-[(2-chloro-4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-propyl-N-(thiophen-3-ylmethyl)acetamide
1-(2-phenoxybenzoyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
1-(2-chlorophenyl)-3-(1-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-[(2-fluorophenyl)methyl]-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-amine
(3S,4R)-3-cyclopropyl-N,N-dimethyl-4-[2-(methylsulfanyl)benzamido]pyrrolidine-1-carboxamide
N,5-dimethyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-2-phenylfuran-3-carboxamide
N-{[1-(pyrrolidin-1-ylmethyl)cyclopropyl]methyl}-4-(4H-1,2,4-triazol-4-yl)benzamide
3-[({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(methyl)amino]-1-phenylpropan-1-ol
2-oxo-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)-1,3-oxazolidine-4-carboxamide
N-ethyl-4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[(5-methylfuran-2-yl)methyl]benzamide
3-methyl-5-(2-{4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(3-hydroxypropyl)-9-(3-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(2-methyl-1-benzothiophen-3-yl)-1H-1,2,3-triazole
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carboxamide
5-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
{1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl}methanamine
methyl 2-[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})carbamoyl]piperidine-1-carboxylate
7-cyclopropanecarbonyl-4-{octahydropyrrolo[1,2-a]piperazin-2-yl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine
(2S,4R)-4-(2-hydroxyacetamido)-N-methyl-1-[(5-phenylthiophen-2-yl)methyl]pyrrolidine-2-carboxamide
{1-[(4-methoxypyridin-2-yl)methyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
N-({5-[(2,3-dimethoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
4-[2-(dimethylamino)-6-oxo-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-8-yl]benzoic acid
1-(2-{4-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)pyrrolidin-2-one
N-[3-({[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl](methyl)carbamoyl}amino)-4-methylphenyl]acetamide
N-(2-hydroxyethyl)-6-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-methyl-3-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1,2,3,4-tetrahydroisoquinoline
2-[4-(5-methoxy-3-methyl-1H-indole-2-carbonyl)-1-methylpiperazin-2-yl]ethan-1-ol
[(2S,6S)-4-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-(3-phenyl-1,2,4-oxadiazol-5-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
5-acetyl-N-(2-phenylethyl)-N-(pyridin-3-ylmethyl)thiophene-3-carboxamide
9-methoxy-3-(2-methoxypyridine-3-carbonyl)-N-methyl-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N3-ethyl-N5-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-{2-[({3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}amino)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}ethan-1-one
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]ethan-1-one
1-[4-(1-benzofuran-2-yl)pyrimidin-2-yl]-5-cyclopropyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
N-{[(2R)-1-ethylpyrrolidin-2-yl]methyl}-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-7-methyl-2-oxo-1H,2H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
[(4-chloro-3-fluorophenyl)methyl](methyl)[(1-methylpyrrolidin-3-yl)methyl]amine
2-{[4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methyl}-5,8-dimethylquinolin-4-ol
2-{3-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]phenoxy}-1-(piperidin-1-yl)ethan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(3S,4R)-1-[(3,5-dichloropyridin-4-yl)methyl]-4-propylpyrrolidin-3-yl]acetamide
dimethyl({2-[5-(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)-1,2,4-oxadiazol-3-yl]ethyl})amine
3-[3-(morpholine-4-carbonyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4,5,6,7-tetrahydro-2H-indazole
3-(hydroxymethyl)-N-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
3-[1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]pyridine