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1-[benzyl(methyl)amino]-3-(4-{[ethyl(methyl)amino]methyl}phenoxy)propan-2-ol
1,6-dimethyl-N-[1-(pyridin-3-yl)pentyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3S,9aR)-8-(4-methylbenzoyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
5-methyl-N4-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)pyrimidine-2,4-diamine
9-[(2R)-2-amino-3-phenylpropanoyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(4-aminoazepan-1-yl)-2-oxoethyl]-3-methoxy-1,2-dihydropyridin-2-one
N-[(3-ethoxyphenyl)methyl]-1-(2-methoxyethyl)-N-(prop-2-en-1-yl)pyrrolidine-3-carboxamide
3-(2-benzyl-5-oxopyrrolidin-2-yl)-N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]propanamide
1-{imidazo[1,2-a]pyridine-3-carbonyl}-4-(2-methoxyphenoxy)piperidine
5-cyclopropanecarbonyl-1'-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-{1-[1-(2-methoxyphenyl)piperidin-4-yl]piperidin-3-yl}-4-(2-methylphenyl)piperazine
(2R,3R,6R)-5-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-phenyl-N-[2-(pyrrolidin-1-yl)ethyl]-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
4-ethoxy-N-[2-(1,3-thiazol-2-yl)ethyl]pyrimidin-2-amine
5-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]-2,8-diazaspiro[4.5]decane
5-(3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
1-[1-({1-[(1-ethyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
2-methyl-5-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,4-dihydropyridin-4-one
2-(2,4-difluorophenyl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}acetamide
2-{1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]pyrrolidin-3-yl}benzoic acid
N-(1-{1-[(2R)-2-aminopropanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
4-[4-(2-{[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}phenoxy)butyl]morpholine
N-{[1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]methyl}adamantane-1-carboxamide
N-methyl-2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]-N-(thian-4-yl)acetamide
3-amino-1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}propan-1-one
2-methyl-7-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}-[1,3]oxazolo[5,4-d]pyrimidine
1-(2-methoxy-5-methylphenyl)-3-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}urea
methyl 1-[2-hydroxy-3-(3-{[methyl(propan-2-yl)amino]methyl}phenoxy)propyl]piperidine-4-carboxylate
4-[(1-{1-[(2-chlorophenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]piperazin-2-one
7-(2-methoxyethyl)-2-[4-(1H-pyrazol-4-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
4-(1H-1,3-benzodiazol-1-yl)-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidine-4-carboxylic acid
methyl 4-{[3-(2-{[(5-methylfuran-2-yl)methyl]carbamoyl}ethyl)piperidin-1-yl]methyl}benzoate
N-[4-({cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenyl]acetamide
3-(2-methylphenyl)-3-[2-(morpholin-4-yl)-2-oxoethyl]-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
N-[2-(4-fluorophenyl)ethyl]-2-(morpholin-3-yl)-N-(pyridin-3-ylmethyl)acetamide
N-[(1-ethyl-1H-indazol-3-yl)methyl]-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[2-(1H-imidazol-1-yl)ethyl]-N-methylpyridin-2-amine
1-ethyl-3-methyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)piperidine-3-carboxamide
5-cyclopropyl-N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-1,2-oxazole-4-carboxamide
N-[(2-chlorophenyl)methyl]-N-(propan-2-yl)-1,4-dioxane-2-carboxamide
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
N-(propan-2-yl)-6-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
N-[(3R,4S)-4-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)pyrrolidin-3-yl]methanesulfonamide
1-[4-(2-methyl-1H-imidazol-1-yl)butan-2-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(3-methoxypropyl)-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(3-methyl-1,2-oxazol-5-yl)methyl]-8-(6-methylpyridin-2-yl)-1,8-diazaspiro[4.5]decane