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(3R,4R)-1-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
(3aR,6aS)-5-{[3-(2-methylphenyl)phenyl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({[2-(piperazin-1-yl)ethyl]amino}methyl)piperidin-2-one
(1R,9aR)-1-[(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)methyl]-octahydro-1H-quinolizin-1-ol
N-(oxolan-2-ylmethyl)-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-amine
3-({4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
2-(dimethylamino)-N,4-dimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]pyrimidine-5-carboxamide
3-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]amino}methyl)-N-(1-methyl-1H-1,2,3-triazol-4-yl)benzamide
3-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}urea
2-(2H-1,3-benzodioxol-5-yl)-1-{3-[5-(2-fluorophenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
3-chloro-N-(1-ethyl-5-oxopyrrolidin-3-yl)-4-fluoro-1-benzothiophene-2-carboxamide
4-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}pyridine
N-ethyl-2-(morpholin-4-yl)-2-(pyridin-3-yl)-N-(pyridin-4-ylmethyl)acetamide
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-3-(1H-pyrazol-1-yl)propanamide
8-(4-methylpentyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(1,2-oxazol-3-ylmethyl)-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
methyl 4-[(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}phenyl)formamido]butanoate
N-[(1R,3R)-3-aminocyclopentyl]-4-methoxy-3,5-dimethylbenzamide
N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}thian-4-amine
5-benzyl-N-(1-ethyl-5-oxopyrrolidin-3-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
8-benzyl-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
ethyl 2-{2-cyclopropyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}acetate
N-(5-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-1-(2-phenylethyl)-1H-1,3-benzodiazol-7-yl)-2-methoxyacetamide
2-(3-methylfuran-2-carbonyl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidine
4-chloro-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
(furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl](pyridin-4-ylmethyl)amine
7-methoxy-N-{3-[methyl(phenyl)amino]propyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1S,5R)-3-[(4-fluoro-3-methoxyphenyl)methyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(4-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperazin-1-yl)quinazoline
5-[4-hydroxy-1-(2-methylpropyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
3-(azetidine-1-sulfonyl)-N-(5-fluoropyridin-3-yl)benzamide
9-[3-(3-hydroxy-3-methylbutyl)benzoyl]-3,9-diazaspiro[5.5]undecane-2,4-dione
4-ethyl-3-{1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{5-[(2-methyl-1H-indol-3-yl)methyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}butan-2-ol
2-amino-6-(2-fluoro-4-hydroxyphenyl)-4-[3-(2-hydroxyethoxy)phenyl]pyridine-3-carbonitrile
2-{4-[6-amino-2-(dimethylamino)pyrimidin-4-yl]-1H-pyrazol-1-yl}-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
3-chloro-4-[(1-cycloheptylpiperidin-4-yl)oxy]-N-(2-methoxyethyl)benzamide
2-methoxy-4-[3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyridine-3-carbonitrile
3-(2-chlorophenyl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-3-phenylpropanamide
3-({3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridin-2-amine
N,N-dimethyl-1-[1-(4,6,7-trimethylquinazolin-2-yl)piperidin-4-yl]pyrrolidin-3-amine
1-(2-aminoethyl)-N-({5,7-dimethylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
(1R,2S,4R)-N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
(5S,9aS,9bS)-5-(2,3-difluorophenyl)-2-(2,3-dihydro-1H-inden-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-benzyl-4-[1-(2-hydroxyethyl)-1H-pyrazol-4-yl]benzene-1-sulfonamide
3-cyclopropyl-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-pyrazole-5-carboxamide
3-[3-cyclopropyl-5-(4-oxo-4-phenylbutyl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
(3aR,6aS)-5-{[3-(cyclopentyloxy)phenyl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(3R,4S)-3-[2-(benzyloxy)acetamido]-4-(propan-2-yl)pyrrolidin-1-yl]propanoic acid