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[(3R,4R)-4-[(dimethylamino)methyl]-1-[4-(piperidin-1-ylmethyl)benzoyl]pyrrolidin-3-yl]methanol
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(4-methyl-1H-pyrrole-2-carbonyl)pyrrolidin-3-yl]methanol
(2S)-2-[({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)amino]-4-methylpentanamide
N-(1,3-benzoxazol-2-ylmethyl)-1-[2-(4-chlorophenyl)ethyl]-N-methyl-6-oxopiperidine-3-carboxamide
2-[3-(propan-2-yloxy)benzoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3,6,7-trimethyl-N-[(1R,2S)-2-phenylcyclopropyl]-1-benzofuran-2-carboxamide
4-(dimethyl-1,2-oxazol-4-yl)-3-(pyridin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-ethyl-3-{1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(but-2-yn-1-yl)-4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridine
6-(4-fluorophenyl)-N,N-dimethyl-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-{[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-(2,5-dihydro-1H-pyrrol-1-ylmethyl)-N-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]benzamide
2-[1-(2-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]pyridin-4-amine
3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1,6-dimethyl-1,2-dihydropyridin-2-one
N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(5-oxopyrrolidin-2-yl)acetamide
(1S,5R)-3-benzyl-6-[(3,4-dimethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
1-(4-ethoxyphenyl)-3-(oxolan-2-ylmethyl)-3-(thiophen-3-ylmethyl)urea
N-(3-hydroxybutyl)-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-amino-6-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-ethyl-4-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
3-hydroxy-3-[({imidazo[1,2-a]pyridin-3-ylmethyl}amino)methyl]-1-(3-phenylpropyl)piperidin-2-one
N-[(6-chloropyridin-3-yl)methyl]-N-methyl-2-(phenylamino)pyrimidine-5-carboxamide
(2R)-2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyrrolidine
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)prop-2-ene-1-sulfonamide
(3S,7S,8aS)-7-{[(2,4-difluorophenyl)methyl]amino}-3-[(1R)-1-hydroxyethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-ethyl-2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
1-methyl-5-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1,2-dihydropyridin-2-one
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]benzamide
5-cyclopropyl-N-[(1-ethylpyrrolidin-2-yl)methyl]-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N,2,4-trimethyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1,3-thiazole-5-carboxamide
2-[3-(3-chloro-4-methoxyphenyl)phenyl]-5-methyl-1,3,4-oxadiazole
{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
2-amino-6-(furan-2-yl)-4-[3-(2-hydroxyethoxy)phenyl]pyridine-3-carbonitrile
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(pyridin-2-yl)piperidine-3-carboxamide
(2R,3R,6R)-5-[(5-ethylfuran-2-yl)methyl]-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
4-(1-ethylpiperidine-2-carbonyl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
2-amino-4-(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)-6-(pyridin-3-yl)pyridine-3-carbonitrile
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
5-methyl-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)-1,2-oxazole-3-carboxamide
(3aS,6aS)-2-[(4-chloro-2-fluorophenyl)methyl]-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2S)-2-amino-1-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(1H-imidazol-4-yl)propan-1-one
1-methyl-5-{1-[2-(thiophen-3-yl)-1H-imidazol-1-yl]propyl}-1H-1,2,4-triazole
(2S)-3-phenyl-2-{[2-(phenylamino)pyrimidin-5-yl]formamido}propanamide
{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amine
2-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]-3,5,7-trimethyl-1H-indole
1-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
8-(1H-imidazol-2-ylmethyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid