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4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-(1,3-thiazole-4-carbonyl)piperidine
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-(pyridin-4-ylsulfanyl)acetamide
3-[(3R,4S)-1-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-(dimethylamino)piperidin-3-yl]propan-1-ol
1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-4-(thian-4-yl)piperazine
5-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]sulfonyl}-2-chloro-4-fluorobenzoic acid
2,3,5-trimethyl-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-[(4-chlorophenyl)methyl]-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-6-oxopiperidine-3-carboxamide
(1R,5R)-6-({[(2-methoxyphenyl)methyl]carbamoyl}methyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
ethyl 1-[2-(methylamino)pyridine-4-amido]cyclobutane-1-carboxylate
N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-2-methylpropanamide
3-methoxy-1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-one
2,3-dimethoxy-N-({1-[3-(methylsulfanyl)propyl]piperidin-3-yl}methyl)benzamide
3-(3-fluorophenyl)-4-[2-(methylamino)pyridine-4-carbonyl]piperazin-2-one
2-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
5-[2-(3-methoxypropyl)-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1R,7S)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-[2-(4-methylphenyl)ethyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(5-methoxyfuran-2-carbonyl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
(1R,5R)-6-(3-methylbut-2-en-1-yl)-3-[4-(1H-pyrazol-3-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[(1-methylpiperidin-3-yl)methyl]benzamide
N,N-dimethyl-2-{4-[1-(pyridin-2-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}acetamide
1-{2-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}-1,4-dihydroquinolin-4-one
(2S)-2-amino-3-(1H-imidazol-4-yl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]propanamide
(3S,4R)-4-methyl-1-[4-(4-methylpiperazin-1-yl)benzoyl]piperidine-3,4-diol
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}propanamide
3-[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-4-yl]-N-(3-chloro-4-fluorophenyl)propanamide
2-(morpholin-4-yl)-N-{[7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(pyridin-3-yl)acetamide
4-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}morpholine
5-methyl-5-phenyl-1-[(1r,4r)-4-hydroxycyclohexyl]piperidin-2-one
6-[4-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
3-(3-fluorophenyl)-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-sulfonamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl]methanol
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-N-(3-ethoxypropyl)propanamide
6-methyl-5-{[3-(2-phenylethyl)piperidin-1-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
8-[3-(difluoromethoxy)benzoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-6-methylimidazo[2,1-b][1,3]thiazole-5-carboxamide
[(3-chloropyridin-4-yl)methyl](methyl)[1-(pyridin-4-yl)ethyl]amine
(1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)(pyridin-2-yl)methanol
N-[1-(pyrrolidin-1-ylmethyl)cyclohexyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
8-(1-methyl-2-oxo-1,2-dihydroquinoline-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-{5-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
6-methyl-2-[({2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}amino)methyl]quinolin-4-ol
2-(dimethylamino)-N,4-dimethyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]pyrimidine-5-carboxamide
6-ethyl-2-(1-methyl-1H-pyrazol-4-yl)-4-(morpholine-4-carbonyl)quinoline
5-fluoro-N,N-dimethyl-2-[4-(pyridin-4-yl)piperazin-1-yl]pyrimidin-4-amine
1'-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]
N-methyl-N-(pyrazin-2-ylmethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(4-chlorophenyl)-5-cyclopropanecarbonyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
8-[(3,4,5-trimethoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-amino-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)acetamide
3-methyl-7-[3-(3-methylphenyl)piperidine-1-carbonyl]-3,4-dihydroquinazolin-4-one