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3-cyclopropyl-1-[4-(oxan-2-ylmethoxy)phenyl]-3-(pyridin-2-ylmethyl)urea
methyl (2S,3S)-2-({4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxyphenyl}formamido)-3-methylpentanoate
2-(5-{[4-(cyclohex-3-en-1-yl)-1H-1,2,3-triazol-1-yl]methyl}-1,2-oxazol-3-yl)pyridine
2-{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]azetidin-3-yl}pyridine
1-cyclopentanecarbonyl-N-(3-hydroxy-3-phenylpropyl)-N-methylpiperidine-4-carboxamide
1-[(4-fluoro-2-methoxyphenyl)methyl]-3-(pyrrolidin-1-yl)piperidine
3-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}benzoic acid
N,N-dimethyl-2-{methyl[(2E)-2-methyl-3-phenylprop-2-en-1-yl]amino}propanamide
2-(2-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}phenoxy)acetic acid
1-cyclohexyl-N-(2-methylpropyl)-4-oxo-5-[4-(thiophene-2-carbonyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
N-[(2,3-dimethoxyphenyl)methyl]-1-(methoxymethyl)cyclopropane-1-carboxamide
3-(4-fluorophenyl)-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
5-ethyl-N-methyl-N-[2-(morpholin-4-yl)propyl]pyrimidin-2-amine
3-(2-amino-1,3-thiazol-4-yl)-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]propan-1-one
{4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1,4-oxazepan-6-yl}methanol
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-2-propyl-1,3-thiazole-4-carboxamide
3-phenyl-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]pyrrolidin-3-ol
2,6-dimethyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}quinoline-4-carboxamide
N-[(2-ethoxypyridin-3-yl)methyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-methyl-4-{[5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)furan-2-yl]methyl}piperazine
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(oxane-4-carbonyl)pyrrolidin-3-yl]acetamide
2-amino-4-(3,4-difluorophenyl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-(5-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyridin-2-yl)acetamide
1-[(2-fluorophenyl)methyl]-6-oxo-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}piperidine-3-carboxamide
3-(3-chlorophenyl)-N-methyl-3-phenyl-N-(pyrazin-2-ylmethyl)propanamide
N-methyl-N-[2-(2-methylpiperidin-1-yl)ethyl]thian-4-amine
2-amino-6-[1-(2-methoxyethyl)-1H-indol-3-yl]-4-(pyridin-3-yl)pyridine-3-carbonitrile
3-(3-hydroxy-3-methylbutyl)-N-[(3R,4R)-4-(4-methylpiperazin-1-yl)oxolan-3-yl]benzamide
(3S,4S)-4-methyl-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidine-3,4-diol
2-(3-fluoropyridin-4-yl)-3-(pyrrolidine-1-carbonyl)pyridine
1-methyl-4-[2-(morpholin-4-yl)-2-oxoethyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
4-[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]benzene-1-sulfonamide
4-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-2-phenylmorpholine
4-[2-(4-cyclopentylphenyl)-5-fluoropyrimidin-4-yl]morpholine
1-(benzyloxy)-8-[1-(pyridin-2-yl)piperidine-3-carbonyl]-1,8-diazaspiro[4.5]decan-2-one
4-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]pyrimidin-2-amine
8-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4aS,8aS)-2-[(2,4-dimethoxy-3-methylphenyl)methyl]-decahydroisoquinolin-4a-ol
(3R,4S)-4-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1,4-diazepan-1-yl)oxolan-3-ol
2-(3-chloro-6-oxo-1,6-dihydropyridazin-1-yl)-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)acetamide
N-ethyl-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-2-(pyridin-2-yl)acetamide
methyl (1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)-1H-pyrrole-2-carboxamide
2-(dimethylamino)-7-(2-methoxybutanoyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-benzyl{[5-chloro-2-(1H-1,2,4-triazol-1-yl)phenyl]amino}sulfonamide
3-methoxy-1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidine
4-methyl-6-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrimidin-2-amine
2-[4-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]pyrrolidine-1-carboxamide
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[(4-phenyloxan-4-yl)methyl]pyrrolidin-2-one