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4-(1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidine-4-carbonyl)morpholine
4-[(2-hydroxyethyl)sulfamoyl]-N-[1-(pyridin-3-yl)propan-2-yl]benzamide
{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
1-methyl-6-{[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methyl}-1H-indole
(4aR,8aR)-2-methanesulfonyl-7-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-decahydro-2,7-naphthyridin-4a-ol
4-[3-(2-methyl-1H-imidazol-1-yl)propyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[5-(methoxymethyl)-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-1-yl]benzoic acid
2-ethoxy-3-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyridine
2-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propane-1,3-diol
methyl 6-[(2-ethoxyphenyl)methyl]-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(3-cyano-2-methyl-1H-indol-1-yl)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}acetamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}benzamide
3-[(1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)oxy]pyridine
methyl 6-({methyl[1-(thiophen-2-yl)ethyl]amino}methyl)-3-(4-methylbenzamido)thieno[2,3-b]pyridine-2-carboxylate
2-methyl-5-{2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine-1-carbonyl}-1H-1,3-benzodiazole
2-methyl-4-(2-methylphenyl)-1-[3-(1H-pyrazol-1-yl)benzoyl]piperazine
2-cyclopropyl-N-methyl-6-oxo-N-[(4-phenoxyphenyl)methyl]-1,6-dihydropyrimidine-5-carboxamide
methyl (2S)-3-methyl-2-[(5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazol-3-yl)formamido]butanoate
1-{3-[(diethylamino)methyl]phenyl}-3-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]urea
2-[1-(2,5-dimethylphenyl)-5-[3-(propan-2-yl)-1,2-oxazol-5-yl]-1H-1,2,4-triazol-3-yl]acetamide
5-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridin-2-amine
5-(3-chloro-4-methoxyphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
methyl 3-[(pyridin-2-ylformamido)methyl]-5-[2-(thiophen-3-yl)acetamido]benzoate
N-{3-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-oxopropyl}-N-methylmethanesulfonamide
(3aS,6aS)-N-(2,4-difluorophenyl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-octahydropyrrolo[2,3-c]pyrrole-5-carboxamide
(1,3-benzothiazol-2-ylmethyl)(methyl){[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
2-{4-[6-amino-5-cyano-4-(furan-3-yl)-3-methylpyridin-2-yl]phenoxy}acetic acid
9-(4-tert-butylbenzenesulfonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
N-(furan-3-ylmethyl)-N,1-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3R,5S)-N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
3-{[1-benzyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]methyl}-3,4-dihydroquinazolin-4-one
3-{[(2S,4S)-4-amino-1-methylpyrrolidin-2-yl]formamido}-N-(2,5-dimethylphenyl)propanamide
4-[(1-acetylpiperidin-4-yl)oxy]-N-[3-(dimethylamino)-2,2-dimethylpropyl]-3-methoxybenzamide
2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-fluoropyridine
2-cyclopropyl-N-[2-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
5-[methyl(2-phenylethyl)amino]-2-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-2,3-dihydropyridazin-3-one
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-5-methyl-1,3,4-oxadiazol-2-amine
3-chloro-4-hydroxy-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
N-[(4-phenylmorpholin-2-yl)methyl]-5-propyl-1,2-oxazole-3-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-(4-ethylphenyl)-5-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-N-[(1S)-1-phenylethyl]pyrimidin-2-amine
N-methyl-3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)propanamide
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}[3-(propan-2-yloxy)propyl]amine
N-(2-hydroxyethyl)-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
3-ethyl-4-methyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-1H-pyrazole-5-carboxamide
4-(2-fluorophenoxy)-1-[3-(methylsulfanyl)propanoyl]piperidine-4-carboxylic acid
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-2,3-dihydro-1-benzofuran-7-carboxamide
2-({4-[2-(furan-2-yl)pyrimidin-5-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)phenol
1-cyclohexyl-N-[(6-hydroxypyrimidin-4-yl)methyl]piperidine-4-carboxamide