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(1R,5R)-N,N-dimethyl-6-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-6-(4H-1,2,4-triazol-4-yl)pyridine
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-5-(1-methyl-1H-pyrazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-[4-(propan-2-yl)phenyl]-1-[1-(1,3-thiazol-2-yl)ethyl]-1H-1,2,3-triazole
6-{1-[2-(1H-imidazol-2-yl)benzoyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
3-cyclopropyl-5-{[(3-methoxyphenyl)sulfanyl]methyl}-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
2-{1-[1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-amine
N-({1-[(3,4-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)-6-oxo-1,6-dihydropyridine-3-carboxamide
1-[3-(difluoromethoxy)benzoyl]-3-(2-methoxyphenoxy)azetidine
[(2S,6S)-4-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
8-[2-(4-fluorophenoxy)acetyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
4-{[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]amino}-N-[(2,3-dimethoxyphenyl)methyl]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-({1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-3-yl}methyl)-4-phenylbenzamide
N-(2-methoxyethyl)-5-methyl-N-[(4-methylphenyl)methyl]pyrazine-2-carboxamide
4-(8-fluoroquinoline-2-carbonyl)-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(dicyclopropylmethyl)piperidine-3-carboxamide
4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazin-2-one
N-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
4-(1-methyl-1H-imidazol-2-yl)-N-[3-(trifluoromethyl)phenyl]piperidine-1-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
1-(2-phenylethyl)-N-{2-[3-(trifluoromethyl)phenyl]ethyl}-1H-1,2,3-triazole-4-carboxamide
N-methyl-N-(pyrazin-2-ylmethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-cyclohexyl-3-(4-fluoro-2-methylphenyl)-1-(pyridin-3-ylmethyl)urea
3-[(2-methoxyethyl)sulfamoyl]-5-(4-methyl-1H-pyrazol-1-yl)benzoic acid
(3aR,7aS)-5-methyl-2-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
3,5-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1,2-oxazole-4-carboxamide
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
ethyl 3-benzyl-1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidine-3-carboxylate
(5R)-5-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]pyrrolidin-2-one
[(2S,6S)-4-[3-(dimethylamino)benzoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
2-(3-fluorophenoxy)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
methyl 4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carboxylate
1-cyclopentyl-5-[5-(methoxymethyl)furan-2-yl]-1H,4H-pyrazolo[3,4-d]imidazole
5-[3-(4-ethylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4-methyl-1,3-oxazole
2-cyclopropyl-9-(2-ethoxyethyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
4-(1-{1-[(4-phenylphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carbonyl)morpholine
N-[3-(3-ethylphenoxy)propyl]-N-methylimidazo[2,1-b][1,3]thiazole-6-carboxamide
2-ethyl-3-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
(2-methoxyethyl)[(4-methylphenyl)methyl]{[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
dimethyl[(2-{[4-(piperidine-1-carbonyl)pyridin-2-yl]oxy}phenyl)methyl]amine
(1R,4S)-2-[2-(pyrimidin-5-yl)pyridine-3-carbonyl]-2-azabicyclo[2.2.1]heptane
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[2-(4-fluorophenyl)azetidin-1-yl]ethan-1-one
5-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1,2-oxazole
methyl 6-[(2E)-3-(2-fluorophenyl)prop-2-enoyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-(5-ethyl-1,3-oxazol-4-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-methyl-7-[5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-5,6,7,8-tetrahydro-2,7-naphthyridine-4-carbonitrile
5-methyl-1-(4-methylphenyl)-4-[4-(methylsulfanyl)benzoyl]piperazin-2-one
5-benzyl-3-(2,3-dihydro-1H-inden-2-yl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
4-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazin-1-yl]pyridine-3-carbonitrile