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1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-3-amine
1-(3-ethyl-1H-pyrazole-4-carbonyl)-2-[2-(thiophen-2-yl)ethyl]piperidine
[7-(5-ethylpyrimidin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methanamine
2-amino-3-ethyl-N-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
8-[(5-chlorofuran-2-yl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-methyl-3-(thiomorpholine-4-carbonyl)-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-(1-hydroxypropan-2-yl)benzamide
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(pyridine-3-carbonyl)pyrrolidin-3-yl]methanol
2-(5-acetylthiophen-3-yl)-1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
5-[4-(thiophen-2-yl)-1H-imidazol-1-yl]pyridin-2-amine
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(5-propylthiophene-3-carbonyl)pyrrolidin-3-yl]methanol
1-[4-(1H-imidazol-4-yl)phenyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
3-ethyl-4-{3-methoxy-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-[(1H-indol-5-ylmethyl)(methyl)amino]-N-methylbutanamide
N-[3-(3-chlorophenyl)phenyl]-1-[2-(pyridin-3-yl)acetyl]piperidine-4-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(2R,3R)-3-{1,5,7-trimethyl-3,7-diazabicyclo[3.3.1]nonan-3-yl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-(methoxymethyl)-6-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}pyrimidine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-(4-fluoro-2-methylphenyl)-3-[1-(quinolin-8-ylmethyl)piperidin-3-yl]propanamide
3-(2-{[ethyl(methyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)propanamide
2-{5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(4-fluorophenoxymethyl)-1H-1,2,4-triazol-1-yl}acetic acid
1-benzyl-5-{[(2-methoxyphenyl)methyl]amino}-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
1-{5-[(4-methyl-3-phenylpiperazin-1-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carbonyl}azocane
1-{[5-(hydroxymethyl)furan-2-yl]methyl}-N-[3-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
5-(3-phenylpropyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
ethyl 2-[({2-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)(methyl)amino]acetate
10-methoxy-5-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
1-{3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}-2-(pyridin-2-ylsulfanyl)ethan-1-one
8-[(2-ethyl-1,3-thiazol-4-yl)methyl]-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
3-(4-hydroxyphenyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1H-pyrazole-5-carboxamide
2-amino-4-{2-[2-(dimethylamino)ethoxy]phenyl}-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
4-{3-cyclopentyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1-ethylpyrrolidin-2-one
(benzylsulfamoyl)(methyl){[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
({5-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
2-[(4-chlorophenyl)methyl]-8-[(1-methylpyrrolidin-3-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
methyl 4-({1-[(2-methoxyphenyl)methyl]-6-oxopiperidin-3-yl}formamido)butanoate
1-ethyl-N-methyl-N-[3-(oxolan-2-yl)propyl]piperidin-4-amine
1-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-2-(methylsulfanyl)ethan-1-one
1-methyl-5-{[2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}piperidin-2-one
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(4-methyl-1H-imidazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-{[5-(3-phenylbutyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}cyclobutanecarboxamide
(3S,4S)-3-hydroxy-4-(morpholin-4-yl)-N-(2,4,6-trimethylpyridin-3-yl)pyrrolidine-1-carboxamide
(3S,4S)-1-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-4-(propan-2-yloxy)pyrrolidin-3-ol
2-cyclopropyl-N-[(4-sulfamoylphenyl)methyl]pyrimidine-5-carboxamide
4-ethyl-3-methyl-5-({2-[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}sulfanyl)-4H-1,2,4-triazole
11-[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one