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2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[3-(morpholin-4-yl)propyl]acetamide
N-cyclopropyl-1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]piperazine-2-carboxamide
2-{3-[hydroxy(phenyl)methyl]-5-[2-(pyridin-3-yl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
(2S,4R)-4-[4-({[(cyclohexylmethyl)carbamoyl](methyl)amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
[(3R,4R)-1-(3,4-dimethoxybenzenesulfonyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
N-ethyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-{[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl](methyl)amino}-1-phenylpropan-1-ol
{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1H-imidazol-5-yl)methyl]amine
N-[(2-chlorophenyl)methyl]-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
2-[(6-{1H-pyrazolo[3,4-b]pyridin-1-yl}quinazolin-4-yl)amino]ethan-1-ol
8-chloro-2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
2-({1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
5-({2-[(2-chlorophenyl)formamido]ethyl}carbamoyl)thiophene-2-carboxylic acid
(2S)-N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(1H-pyrazole-3-carbonyl)pyrrolidine-2-carboxamide
N-{[1-(dimethylamino)cyclohexyl]methyl}-6-methyl-4-oxo-4H-pyran-2-carboxamide
4-ethyl-2-methyl-6-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidine
(2S,4R)-4-amino-1-[2-(3,5-dimethoxyphenyl)acetyl]-N,N-diethylpyrrolidine-2-carboxamide
1-{5-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]thiophen-2-yl}ethan-1-one
1-[(3-methoxyphenyl)methyl]-N3-[(4-methylphenyl)methyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(2R,3R,6R)-5-(6-methoxypyrimidin-4-yl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(2-{1-[2-(naphthalen-1-yl)ethyl]-1,2,5,6-tetrahydropyridin-3-yl}ethyl)acetamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1H-pyrazole-3-carboxamide
N-(cyclopropylmethyl)-2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]-N-propylacetamide
1-(4-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-2-methoxyphenoxy)-3-(4-ethylpiperazin-1-yl)propan-2-ol
(4aS,8aR)-1-(carboxymethyl)-6-[(3-hydroxyphenyl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
2-{2-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,3-benzodiazole
methyl (2S,4R)-1-{[1-(2-carbamoylethyl)-1H-indol-3-yl]methyl}-4-hydroxypyrrolidine-2-carboxylate
methyl[3-(1H-pyrazol-1-yl)propyl][(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amine
(2S,4R)-4-(4-{[(2-methoxyphenyl)formamido]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
N-[3-(dimethylamino)propyl]-N-methyl-1-[(3,4,5-trimethoxyphenyl)methyl]piperidin-3-amine
3-[4-(4-chloro-1-methyl-1H-indazol-3-yl)-1H-1,2,3-triazol-1-yl]pyrrolidin-2-one
7-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-2-(1,2-oxazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline
3-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-6-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-(1,1-dioxo-1λ6-thian-4-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
(2S)-2-({2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxyphenyl}formamido)propanamide
2-[4-methyl-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-3-yl]-N-pentylacetamide
2,5-dimethyl-3-{4-[3-(pyridin-4-yl)propyl]piperazin-1-yl}pyrazine
1-(4-{5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)-2-(thiophen-3-yl)ethan-1-one
3-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-2-methylphenyl)urea
[(dimethyl-1,3-thiazol-5-yl)methyl](methyl)[(3-methylpyridin-2-yl)methyl]amine
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]pyrrolidin-3-yl]methanol
3-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-(furan-2-ylmethyl)piperidine
5-(5-chloropyrimidin-2-yl)isoquinoline
2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine
1-(6-aminopyrimidin-4-yl)-4-(cyclobutylmethyl)-1,4-diazepane-6-carboxylic acid
3-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroisoquinolin-1-one
1-[6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
2-(1-{2-[(4-benzylpiperazin-1-yl)methyl]-1,3-oxazol-4-yl}-N-methylformamido)-N-methylacetamide
1-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
4-{[1-(carbamoylmethyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide