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4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-N-[1-(pyrimidin-4-yl)ethyl]benzamide
N-(3-methylcinnolin-5-yl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
6-[4-(2-hydroxyethyl)piperazin-1-yl]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
(1S,5R)-6-(2,6-difluoro-4-methoxybenzoyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-(1-{[4-(hydroxymethyl)oxan-4-yl]methyl}-1H-imidazol-2-yl)benzonitrile
3-({[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}methyl)-2-methoxy-6-(propan-2-yl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
4-{[({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}-2-methoxyphenol
1-(pyridin-3-ylmethyl)-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
6-methyl-3-(4-methylpiperazine-1-carbonyl)-1-(oxolan-2-ylmethyl)-2-(2-phenylethyl)-1,4-dihydropyridin-4-one
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
2-(4-acetylpiperazin-1-yl)-N-[(4-acetamidophenyl)methyl]acetamide
2-(1H-1,3-benzodiazol-1-yl)-N-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)acetamide
1,3-dimethyl-N-(2-{4-[(4-phenylpiperidin-1-yl)methyl]phenoxy}propyl)-1H-pyrazole-5-carboxamide
1-ethyl-5-(ethylamino)-N-(furan-3-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-{2-[4-(4-methoxypyrimidin-2-yl)piperazin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonitrile
6-chloro-2-{1-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
5-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
5-(3-methoxyphenoxymethyl)-N-[(3S)-2-oxoazepan-3-yl]-1,2-oxazole-3-carboxamide
N-({5-[(4-ethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
dimethyl[(5-{[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}thiophen-3-yl)methyl]amine
2-(2,5-dioxoimidazolidin-1-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
(3S,4S)-4-(naphthalen-2-yl)-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidin-3-ol
5-acetyl-N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)thiophene-3-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(4-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-6-methylpyridine-3-carbonitrile
4-(carbamoylmethoxy)-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)benzamide
N-({1-[(4,6-dimethylpyrimidin-2-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)thiophene-2-carboxamide
5-[(4-methanesulfonylphenyl)methyl]-3-methyl-1-(3-methylphenyl)-1H-1,2,4-triazole
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(1,2-oxazol-3-ylmethyl)acetamide
2-amino-4-(4-hydroxyphenyl)-6-(3,4,5-trimethoxyphenyl)pyridine-3-carbonitrile
[3-(cyclopropylmethyl)-1-[1-(pyridine-2-carbonyl)piperidin-4-yl]piperidin-3-yl]methanol
2-methyl-8-(5-methylpyrimidin-2-yl)-2,8-diazaspiro[5.5]undecane
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-pyrazole-3-carboxamide
5-(3-acetylphenoxymethyl)-N-[(1-ethylpyrrolidin-2-yl)methyl]-1,2-oxazole-3-carboxamide
1-(2-ethylphenyl)-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazine
1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)acetamide
1-(2-methoxyphenyl)-2,2-dimethyl-4-(3-propyl-1H-pyrazole-4-carbonyl)piperazine
ethyl[(4-ethylphenyl)methyl][(2-methyl-1H-imidazol-4-yl)methyl]amine
3-methyl-6-{5-[3-(2-methylpropyl)-1,2-oxazol-5-yl]-1,2,4-oxadiazol-3-yl}pyridazine
N-[2-(dimethylamino)-2-(4-methylphenyl)ethyl]-4-(trifluoromethyl)pyrimidin-2-amine
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-1-(2-phenylethyl)piperidin-4-amine
1-(2-hydroxy-5-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)ethan-1-one
5-(4-carboxybutanoyl)-1-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazine
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5,6-dimethylpyrimidin-4-amine
7-(cyclopropylmethyl)-2-(4-propoxybenzoyl)-2,7-diazaspiro[4.5]decan-6-one
1'-(pyridin-4-ylmethyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one