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1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-[(3-methylphenyl)methyl]piperazine
[3-(1H-imidazol-1-yl)propyl][(6-methylpyridin-2-yl)methyl](pyridin-4-ylmethyl)amine
1-benzyl-5-{3-methyl-5H,6H-imidazo[2,1-b][1,3]thiazol-2-yl}-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
(2S,4S)-N-ethyl-1-[3-(methylsulfanyl)propanoyl]-4-[2-(pyridin-3-yl)acetamido]pyrrolidine-2-carboxamide
2-(3-methoxypropyl)-8-[2-(morpholin-4-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
1-ethyl-5-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-imidazol-2-yl)-1H-1,2,4-triazole
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-2,3-dihydro-1,4-benzodioxine-6-sulfonamide
1-[2-(piperidin-1-ylmethyl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-[(4-acetyl-4-phenylpiperidin-1-yl)methyl]-1-methyl-1H-pyrrole-2-carbonitrile
5-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
N-(2,5-dimethylphenyl)-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
9-(2-oxoimidazolidine-4-carbonyl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
4-methyl-7-({[(5-methyl-1,2,4-oxadiazol-3-yl)methyl](propan-2-yl)amino}methyl)-2H-chromen-2-one
5-[1-(5-cyclopropyl-4-phenyl-1H-imidazol-1-yl)ethyl]-1-propyl-1H-1,2,4-triazole
2-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
N-methyl-2-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-(propan-2-yl)acetamide
2-methoxy-1-[1'-(oxane-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-(2,3-dihydro-1H-inden-2-yl)-3-[(oxolan-3-yl)sulfamoyl]benzamide
3-({[1-(2-cyclohexylethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}(methyl)amino)propanamide
1-ethyl-5-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-3-(2-methylpropyl)-1H-pyrazole
1-(naphthalen-1-ylmethyl)-N-{1-oxaspiro[4.4]nonan-3-yl}-1H-1,2,3-triazole-4-carboxamide
5-cyclopropyl-1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
N4-ethyl-N2-methyl-N2-[(3-methylpyridin-4-yl)methyl]pyrimidine-2,4-diamine
8-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(azepan-1-yl)propyl]-N-methyl-4-(piperidin-3-yl)benzamide
N-[2-(2-chlorophenyl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3R,4R)-3-cyclopropyl-3-hydroxy-4-methyl-N-[(4-methylphenyl)methyl]pyrrolidine-1-carboxamide
N-{[2-(4-fluorophenyl)-6-methylquinolin-3-yl]methyl}-2,2-dimethyloxan-4-amine
N-[(3R,4R)-1-[3-(benzyloxy)propyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
N-benzyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
3-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-indazole
N-ethyl-5-[(4-methylpiperazin-1-yl)methyl]-N-[(2E)-3-phenylprop-2-en-1-yl]furan-2-carboxamide
2-(1-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}piperidin-2-yl)pyridine
1-[(butan-2-yl)amino]-3-(2,4-dimethylphenoxy)propan-2-ol
1-[1'-(1H-1,3-benzodiazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
({4-ethyl-5-[1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
2-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
(3R,5S)-N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
ethyl (4aS,8aR)-6-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-decahydro-1,6-naphthyridine-4a-carboxylate
1-(4-ethylpiperazin-1-yl)-3-(2-methoxy-4-{[methyl(2-methylpropyl)amino]methyl}phenoxy)propan-2-ol
1-(2-{1-[(2-chloro-6-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}ethyl)-1,2-dihydropyridin-2-one
2-methyl-8-(1-methyl-4-phenylpiperidine-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl]-N,1-dimethyl-3-propyl-1H-pyrazole-5-carboxamide
1-(prop-2-en-1-yl)-N-(propan-2-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(3-methoxybenzenesulfonyl)-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
N-[(3-chlorophenyl)methyl]-3-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}propanamide
3-(5-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,4-triazol-3-yl)pyridine
ethyl 3-[(4-fluorophenyl)methyl]-1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperidine-3-carboxylate