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2-{3-[4-(hydroxymethyl)piperidin-1-yl]piperidine-1-carbonyl}-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
N-[(3-methylphenyl)methyl]-2-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)acetamido]benzamide
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-4-[(3-fluorophenyl)methyl]piperazine
N-(1,2-oxazol-3-ylmethyl)-4-(piperidin-3-yl)benzamide
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1,2-oxazole-3-carboxamide
3-methyl-5-{2-oxo-2-[3-(pyridine-2-carbonyl)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(2-{[3-(3-hydroxypiperidin-1-yl)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
4-chloro-5-[({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-N,N-dimethyl-1,3-thiazol-2-amine
N-cyclopropyl-4-[3-(1-methoxyethyl)phenyl]benzamide
ethyl 3-[(3-chlorophenyl)methyl]-1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidine-3-carboxylate
1-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-3-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-[2-(1H-imidazol-4-yl)ethyl]quinoxaline-5-carboxamide
N'-(2-ethoxyphenyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]propanediamide
N-methyl-N-[2-(oxan-4-yl)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
2-ethyl-N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]pyrimidine-5-carboxamide
4-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}butanamide
(3R,5S)-5-[(4-methylpiperazin-1-yl)methyl]-N-(oxolan-2-ylmethyl)-1-(2-phenylethyl)piperidine-3-carboxamide
1-cyclohexyl-6-(pyridin-3-ylmethoxy)-4-(pyridin-4-ylmethyl)-1,4-diazepan-2-one
N-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}-1-methylpiperidin-4-amine
ethyl 2-chloro-5-({[3-(morpholin-4-yl)propyl]carbamoyl}amino)benzoate
1-(adamantan-2-yl)-4-[(2S,4S)-1-[(3-fluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]piperazine
N-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-6-(piperidin-4-yl)pyrimidin-4-amine
1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(3-methylphenoxy)piperidine
1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-4-(thiophene-2-carbonyl)piperazine
N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-[2-(dimethylamino)ethyl]-3-(4-methylphenyl)propanamide
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]pyridine-2-carboxamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-3-fluorobenzene-1-sulfonamide
N-[(5-chloro-2-propoxyphenyl)methyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
(1R,3S)-3-(2-aminoethoxy)-7-[(2-methoxynaphthalen-1-yl)methyl]-7-azaspiro[3.5]nonan-1-ol
5-{3-oxo-3-[4-(quinazolin-4-yl)piperazin-1-yl]propyl}imidazolidine-2,4-dione
methyl 3-({2-[(quinolin-8-yloxy)methyl]-1,3-oxazol-4-yl}formamido)propanoate
N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-{2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}benzamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]propan-1-one
2-{[1-(2,3-dihydro-1H-inden-5-yl)piperidin-4-yl]amino}-N,N-dimethylethane-1-sulfonamide
N-(cyclopropylmethyl)-3-(4-methylphenyl)-N-propyl-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
2,4-dimethyl-1-({3-[4-(piperidin-1-yl)butoxy]phenyl}methyl)-1,4-diazepane
1-methyl-1'-[(1-propyl-1H-imidazol-2-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-(4-methoxyphenyl)-4-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)piperazine
(1R,7S)-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-4-oxo-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
7-fluoro-N,N-dimethyl-2-{2-[(pyridin-3-ylmethyl)amino]pyrimidin-5-yl}quinoline-4-carboxamide
3-{2-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-oxoethyl}-4-[(2-fluorophenyl)methyl]piperazin-2-one
N-methyl-4-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}pyridin-2-amine
N,N-dimethyl-7-(4-methyl-1H-imidazole-2-carbonyl)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[2-(dimethylamino)ethyl]-4-(3-phenoxyazetidine-1-carbonyl)pyrrolidin-2-one
5-(2-chlorophenyl)-2,4-dimethoxypyrimidine
2-(cyclopropylmethyl)-8-[2-(3,4-dimethylphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
methyl (2S,4S,5R)-5-(2,3-difluorophenyl)-4-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]carbamoyl}-1-methylpyrrolidine-2-carboxylate
4-({5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1,2,4-oxadiazol-3-yl}methyl)morpholine