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N-(2,3-dihydro-1H-inden-2-yl)-N,5-dimethyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
7-[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazole-4-carbonyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{5-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1H-pyrazol-3-yl}phenol
2-methyl-4-(5-{[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}thiophen-2-yl)but-3-yn-2-ol
2-amino-4-(2-ethylpyrimidin-5-yl)-6-(pyridin-2-ylmethyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-(5-acetylthiophen-3-yl)-N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)acetamide
(1R,2R,4R)-N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
[3-(dimethyl-1,2-oxazol-4-yl)propyl]({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl})amine
N-{[1-(cyclohex-2-en-1-yl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}-2,4,6-trimethylbenzamide
methyl 3-[(3S,4R)-1-{[4-(benzyloxy)phenyl]methyl}-4-(morpholin-4-yl)piperidin-3-yl]propanoate
5-{[methyl({5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl})amino]methyl}pyrimidin-2-amine
7-{2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-(2-{1-[2-(2H-1,3-benzodioxol-5-yloxy)propanoyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(propan-2-yloxy)ethyl]acetamide
4-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-1H-imidazole-5-carboxamide
methyl({[1-(morpholin-4-yl)cyclohexyl]methyl}){4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
3-(2-ethyl-1H-imidazol-1-yl)-1-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}propan-1-one
2-[2-(3-methoxypropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]-6-methylpyridine-3-carboxylic acid
1-methyl-4-{2-[4-phenyl-5-(5-propylfuran-2-yl)-1H-imidazol-1-yl]ethyl}piperazine
1-(5-{[bis(prop-2-en-1-yl)amino]methyl}-2-methoxyphenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
1-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
4-({[1-(hydroxymethyl)cyclopentyl]amino}methyl)-2,6-dimethylphenyl acetate
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
2-[7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
7-methyl-4-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-3,4-dihydro-2H-1,4-benzothiazin-3-one
1-cyclopentanecarbonyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}piperidine-4-carboxamide
N,6-dimethyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(pyridin-3-yl)pyrimidin-4-amine
3-(4-methyl-1,3-thiazol-5-yl)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propan-1-one
5-fluoro-2-(1-{imidazo[1,2-a]pyrimidine-2-carbonyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
1-[(3S,4R)-3-cyclopropyl-4-{[6-(methoxymethyl)pyrimidin-4-yl]amino}pyrrolidin-1-yl]-3-methylbut-2-en-1-one
1-({5-[1-(3-methoxypropyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
1-(3,4-difluorophenyl)-5-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}-1H-1,2,4-triazole
5-methyl-N-(1,2-oxazol-3-ylmethyl)-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
methyl 5-[1-(5-methylpyridin-2-yl)propan-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
1-(3,3-diphenylpiperidine-1-carbonyl)cyclopropan-1-amine
N-(cyclopropylmethyl)-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-butyl-1-methyl-4-(7-methyl-1-benzofuran-2-carbonyl)piperazin-2-one
3-methoxy-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]pyrrolidine
5-{3-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
N-cyclooctyl-1-ethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{[4-(1-methanesulfonylpyrrolidin-3-yl)piperidin-1-yl]methyl}pyridine
3-ethyl-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-1H-pyrazole-4-carboxamide
2-(2,4-difluorophenoxy)-1-[4-(dimethylamino)azepan-1-yl]ethan-1-one
(2-methoxyethyl)[(3-methylthiophen-2-yl)methyl]{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
2-[4-(4-cyanophenyl)-3-oxopiperazin-1-yl]-N-[(2-methylphenyl)methyl]acetamide
4-(5-tert-butyl-1H-pyrazol-3-yl)-1-(furan-3-ylmethyl)-1H-1,2,3-triazole
N-[2-hydroxy-2-(pyridin-4-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
4-[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]-4-oxobutane-1-sulfonamide
2-(1-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidine-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline
(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl](pyridin-4-ylmethyl)amine