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2-(2-methyl-1,3-thiazol-4-yl)-N-[(2-propyl-1,3-thiazol-4-yl)methyl]acetamide
3-chloro-6-[4-(2-methylphenoxy)piperidin-1-yl]pyridine-2-carboxylic acid
(3S,5R)-5-[(4-fluorophenyl)carbamoyl]-1-(thiophen-3-ylmethyl)piperidine-3-carboxylic acid
2-[1-(furan-3-ylmethyl)-4-(2-methyl-1,3-thiazole-4-carbonyl)piperazin-2-yl]ethan-1-ol
(4aS,8aR)-1-(3-hydroxypropyl)-6-(pyrrolidine-1-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-(3-acetylpiperidin-1-yl)-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
1-(1-cyclobutanecarbonylpiperidin-4-yl)-2-[2-(2-methoxyphenyl)ethyl]-1H-1,3-benzodiazole
4-[3-phenyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-2-(propan-2-yl)pyrimidine
3-cyclobutyl-4-[4-(dimethylamino)phenyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
N-(4-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}phenyl)acetamide
6-{2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
6-[(diethylamino)methyl]-N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
2-(cyclopentylmethyl)-N,N-diethyl-6-methyl-4-oxo-1-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
3-(4-benzyl-1H-pyrazol-5-yl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
1-methyl-2-(morpholin-4-yl)-5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-1,3-benzodiazole
1-(2-methoxyacetyl)-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
(1R,5R)-6-benzyl-3-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
2-{[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(2-fluorophenyl)ethyl)piperidin-1-yl]methyl}-4-methoxyphenol
(3R,4R)-1-(3-chlorothiophene-2-carbonyl)-3-cyclobutyl-4-methylpyrrolidin-3-ol
5-{[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2-methyl-1,3-thiazole
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-propanoyl-2,7-diazaspiro[4.5]decan-6-one
6-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)pyridine-3-carboxamide
3-(2-{[cyclohexyl(methyl)amino]methyl}phenyl)-1-[2-(6-hydroxypyrimidin-4-yl)ethyl]urea
2-amino-4-(2,3-difluoro-6-methoxyphenyl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
(4S)-3,3,4-trimethyl-1-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}piperidin-4-ol
(2R)-2-amino-3-hydroxy-1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}propan-1-one
N-[3-(3,5-dimethylphenoxy)propyl]-3,5-difluoro-N-methylpyridine-2-carboxamide
2-{methyl[2-(pyridin-2-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1,3-dimethyl-4-{7-methyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carbonyl}piperazin-2-one
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]acetamide
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(2-methoxyethoxy)ethan-1-one
1-ethyl-4-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
1-(2H-1,3-benzodioxol-5-yl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}urea
N-(1-benzyl-1H-pyrazol-3-yl)-2-[4-(2-methoxyphenyl)-1H-pyrazol-1-yl]acetamide
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
3-hydroxy-3-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
3-benzyl-8-[4-(1H-indol-3-yl)butan-2-yl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 1-(2-chloropyridine-4-carbonyl)-3-(2-phenylethyl)piperidine-3-carboxylate
2-phenyl-N-(2,2,2-trifluoroethyl)imidazo[1,2-a]pyridine-6-carboxamide
3-(4-hydroxyphenyl)-2-phenyl-N-(2,2,2-trifluoroethyl)propanamide
1-[(2-methyl-1H-imidazol-4-yl)methyl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
(2S,4S)-4-amino-1-{3-[(4-methylpyridin-2-yl)carbamoyl]propanoyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-methyl-6-[(1-propyl-1H-imidazol-2-yl)methyl]-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
1-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-2-(3-fluorophenyl)ethan-1-one
3-[3-(cyclopentylcarbamoyl)-N-(1-phenylethyl)propanamido]propanoic acid
3-(4-methyl-1,3-thiazol-5-yl)-N-[2-(4-phenylpyrimidin-2-yl)ethyl]propanamide
5-fluoro-N,N-dimethyl-2-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidin-4-amine
(1R,2S,9R)-11-(3,4-dimethoxybenzoyl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}acetamide