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N-[(3S,4R)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
4-cyano-N-[(3R,4S)-1-(1H-imidazol-4-ylmethyl)-4-propylpyrrolidin-3-yl]oxane-4-carboxamide
2-[(4-chlorophenyl)methanesulfonyl]-2,7-diazaspiro[4.5]decane
4-[7-(1-phenylcyclopentanecarbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
5-fluoro-2-(1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
3-[(3R,4S)-1-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
2-({[(3R,4R)-4-(hydroxymethyl)-1-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(ethanesulfonyl)piperidine-3-carboxylate
6-{2-[5-(1-ethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyrimidin-4-ol
4-[1-(cyclohex-3-ene-1-carbonyl)piperidin-3-yl]-5-methyl-2-[(pyridin-2-ylmethyl)sulfanyl]pyrimidine
3-[(3aS,6aS)-octahydropyrrolo[3,4-b]pyrrole-5-sulfonyl]-N-(pyridin-3-yl)benzamide
4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}-1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine
N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-{[2-(pyrrolidin-1-yl)ethyl]amino}pyridine-3-carboxamide
(3aR,6aS)-2-(cyclopropylmethyl)-5-(4-methoxybenzoyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-methoxyethyl)-6-oxo-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]piperidine-3-carboxamide
4-[2-(1,4-oxazepan-4-yl)-2-oxoethyl]-1-phenyl-3-propyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aS,7aR)-N-(2,5-dimethylphenyl)-6,6-dioxo-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-cycloheptyl-3-[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]propanamide
3-(3-methoxyphenyl)-4-[3-(propan-2-yl)-1,2-oxazol-5-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-({4-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)acetic acid
N-cyclobutyl-2-(dimethylamino)-2-(2-fluorophenyl)acetamide
1-[4-({[(2-methoxyphenyl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
6-(3-hydroxyphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
8-{[2-(trifluoromethyl)phenyl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
N,2-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-(furan-2-ylmethyl)-1-[6-(methoxymethyl)pyridine-2-carbonyl]piperidine-4-carboxamide
N-[2-(6-hydroxypyrimidin-4-yl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
N-[(3S,4R)-1-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
ethyl 1-(2-hydroxyethyl)-5-(quinoxalin-5-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
8-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}acetyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-amino-4-(2-ethylpyrimidin-5-yl)-6-(5-methylfuran-2-yl)pyridine-3-carbonitrile
N-[2-(4-methoxyphenyl)phenyl]-1-[(2-methylpyrimidin-5-yl)methyl]pyrrolidine-2-carboxamide
1-{4-[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]phenyl}pyrrolidin-2-one
2-[(oxolan-2-ylmethyl)amino]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-(pyridin-2-yl)pyrimidin-2-amine
1-[(4-fluorophenyl)methyl]-5-[4-(propan-2-yl)benzoyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
2,2-dimethyl-1-{4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}butan-1-one
3-(dimethylamino)-N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)benzamide
6-[(diethylamino)methyl]-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-(furan-2-ylmethyl)-1-(pyrazin-2-yl)piperidine-4-carboxamide
(3R,4S)-1-[1-(4-fluoro-2-methylphenyl)piperidin-4-yl]-3,4-dimethylpiperidin-4-ol
5-methanesulfonyl-N-(3-methylbutyl)-4-(piperidin-3-yl)pyrimidin-2-amine
1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
3-{[(furan-2-ylmethyl)amino]methyl}-6,7-dimethoxy-1-[(4-methylphenyl)methyl]-1,2-dihydroquinolin-2-one
2-[3-(oxan-4-yl)-5-(pyrazin-2-yl)-1H-1,2,4-triazol-1-yl]acetic acid
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(pyridin-3-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
2-{[(2,3-dihydro-1H-inden-2-yl)(methyl)amino]methyl}-6-methoxyphenol
(1S,5R)-3-benzyl-6-(3,5-difluoropyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-{2-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]pyrimidin-4-yl}pyrrolidin-3-ol