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2-{1-[8-chloro-2-(furan-2-yl)quinoline-4-carbonyl]pyrrolidin-2-yl}ethan-1-ol
4-methyl-N-[2-(N-methylmethanesulfonamido)ethyl]-2-(4-methylpiperazin-1-yl)pyrimidine-5-carboxamide
4-ethyl-3-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(5-methyl-1H-pyrazol-1-yl)acetamide
1-(2-propyl-1,3-thiazole-4-carbonyl)-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
5-(1H-imidazol-1-ylmethyl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]furan-2-carboxamide
N-{3-[4-(4-methylphenyl)-2-(morpholin-4-yl)pyrimidin-5-yl]phenyl}acetamide
N-methyl-6-oxo-N-(2-phenoxyethyl)-1,6-dihydropyridine-3-carboxamide
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(pyrrolidin-3-yl)benzamide
(4aS,8aR)-1-(3-methoxypropyl)-6-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-decahydro-1,6-naphthyridin-2-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
2-hydroxy-4-methyl-1-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]pentan-1-one
2-(2-hydroxyethyl)-8-(2,4,5-trimethylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
8-[4-(1H-1,2,4-triazol-1-yl)phenyl]-1H,2H,5H,6H,7H,8H-[1,3]oxazolo[4,5-g]quinoline-2,6-dione
3-{2-oxo-4-[3-(1H-pyrazol-1-yl)butanoyl]piperazin-1-yl}benzonitrile
2-[(3-methoxyphenyl)sulfanyl]-N-methyl-N-(quinolin-5-ylmethyl)acetamide
1-(2-{methyl[2-methyl-6-(piperidin-3-yl)pyrimidin-4-yl]amino}ethyl)piperidin-2-one
2-cyclohexyl-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-[benzyl(1H-imidazol-4-ylmethyl)amino]-2-methylpropan-1-ol
4-{[3-(4-methoxyphenoxymethyl)piperidin-1-yl]methyl}pyridine
N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
2-(2-{[3-(2-methyl-1H-imidazol-1-yl)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-cyclopropyl-4-propyl-N-(thiophen-3-ylmethyl)pyrimidine-5-carboxamide
2-amino-1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-4-(methylsulfanyl)benzamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-cyclopentylpyrimidin-2-amine
N-{1-[(2-methylphenyl)methyl]cyclopropyl}-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
7-(5-chloropyridin-2-yl)-4-(1,3-thiazol-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{1-[1-(thiophen-2-ylmethyl)piperidin-4-yl]ethyl}morpholine
1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-4-(pyrrolidin-1-yl)pentan-1-one
N2-methyl-N5-[3-(propan-2-yloxy)phenyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2,5-dicarboxamide
2-chloro-N-{[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]methyl}benzamide
(4aS,7aR)-1-[3-(2-methoxyphenyl)propanoyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(2-chloro-4,5-difluorophenyl)ethan-1-one
1-ethyl-2-({1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1H-imidazole
1-cyclopropyl-3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-3-(4-phenylphenyl)pyrrolidine-2,5-dione
3-(2-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}-2-oxoethyl)-5,5-dimethylimidazolidine-2,4-dione
2-(4-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}piperidin-1-yl)pyridine-4-carbonitrile
N-(4-{1-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-1H-imidazol-2-yl}phenyl)acetamide
5-acetyl-6-methyl-3-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-1,2-dihydropyridin-2-one
5-phenyl-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-3-carboxamide
N-{4-methyl-3-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]phenyl}cyclopentanecarboxamide
(1R,2R,6S,7S)-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-4-azatricyclo[5.2.1.02,6]decane
N-[(3,4-difluorophenyl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(4-methyl-1,3-thiazol-5-yl)-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]propan-1-one
6-tert-butyl-3-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
N-[(3S)-1-benzylpyrrolidin-3-yl]-N-methyl-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
N,N-dimethyl-2-[({3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}amino)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
4-[3-(4,4-difluoropiperidine-1-carbonyl)phenyl]-2-methylbutan-2-ol