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N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
3-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-1-{4-[(E)-2-(pyridin-2-yl)ethenyl]phenyl}urea
N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(1H-pyrazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
1-[1-(1-benzothiophen-2-ylmethyl)piperidin-3-yl]-4-phenylpiperazine
3-{1-[2-(2,3-dimethylphenoxy)ethyl]azetidin-3-yl}pyridine
4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-{thieno[3,2-d]pyrimidin-4-yl}piperidine
ethyl 4-{[1-(ethylcarbamoyl)ethyl]amino}piperidine-1-carboxylate
1-benzyl-3-(pyridin-2-ylmethyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(furan-2-ylmethyl)-N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}piperidine-4-carboxamide
1-[3-(1H-pyrazol-1-yl)propyl]-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
1-[(2-fluorophenyl)methyl]-5-[4-(2-hydroxyethyl)piperidine-1-carbonyl]piperidin-2-one
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
3-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
4-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-6-methoxypyrimidin-2-amine
N-[3-(dimethylamino)-1-phenylpropyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
(3R,4S)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-4-cyclopropylpyrrolidin-3-amine
8-chloro-2-[3-(3-methoxypropyl)piperidine-1-carbonyl]quinoline
N,1,3-trimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1-{[methyl({[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl})amino]methyl}cyclopropyl)methanol
7-fluoro-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}quinazolin-4-amine
[3-({1-[2-(methylamino)-1,3-thiazole-4-carbonyl]pyrrolidin-3-yl}methyl)phenyl]methanol
6-methyl-4-[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
4-(2-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}-2-oxoethyl)piperazin-2-one
3-methyl-N-({5-[(oxolan-2-ylmethyl)sulfanyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)thiophene-2-carboxamide
(1S,6R)-9-[2-oxo-8-(prop-2-en-1-yl)-2H-chromene-3-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
(2E)-1-[4-(2-ethyl-5-fluoro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]-3-(4-methoxyphenyl)prop-2-en-1-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-2-methyl-1H-1,3-benzodiazole
(2S)-1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxamide
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-(2,5-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-sulfonyl]-N-(3-methylbutyl)benzamide
1-[9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2-(2-aminoethyl)-N-(cyclopropylmethyl)-N-(2-methoxyethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)pyrimidin-2-amine
2-[(1R,5R)-3-azabicyclo[3.3.1]nonane-3-carbonyl]-6-fluoro-1H-1,3-benzodiazole
N-(3-cyclopentylpropyl)-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-{[(3-hydroxy-2-oxo-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]amino}-N,N-dimethylpropanamide
5-[2-(4-chloro-2-methylphenoxy)acetyl]-N-cyclopentyl-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(1,3-benzothiazol-2-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}propanamide
N-[2-(7-methyl-1H-indol-3-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
cyclopentyl 4-{[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]amino}benzoate
1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}cyclopentan-1-ol
N-cyclohexyl-1-(propan-2-yl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
N-ethyl-2-({methyl[(5-methylthiophen-2-yl)methyl]amino}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
3-chloro-N-cyclopentyl-4-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]oxy}benzamide
8-[3-(3-methoxyphenyl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
N-{2-[(3R)-3-hydroxypyrrolidine-1-carbonyl]-4-methylphenyl}-2-methylpropanamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-{[(2R)-2-carbamoylpyrrolidin-1-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
3-methyl-7-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-(1-methyl-3-phenyl-1H-pyrazol-5-yl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]urea