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5-{[2-(morpholin-4-yl)ethyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
3-(1-{[3-(cyclopentyloxy)phenyl]methyl}piperidin-4-yl)-N-(2-methoxyethyl)propanamide
(4aS,7aR)-1-{2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetyl}-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-(1-ethyl-5-oxopyrrolidin-3-yl)-2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
2-{5-[(benzyloxy)methyl]-1-cyclohexyl-1H-1,2,4-triazol-3-yl}acetamide
5-(2-methoxyphenoxymethyl)-N-(2-phenylethyl)-1H-pyrazole-3-carboxamide
N-(2-hydroxyethyl)-2,6-dimethoxy-N-[(2E)-3-phenylprop-2-en-1-yl]pyrimidine-4-carboxamide
7-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)-1-[(1R,2S)-2-propylcyclopropanecarbonyl]piperidine
1-(1-cyclobutanecarbonylpiperidine-4-carbonyl)-4-phenylpiperidin-4-ol
2-(1-{4-[(benzyloxy)methyl]-1H-1,2,3-triazol-1-yl}ethyl)-1H-1,3-benzodiazole
2-{[5-(2,2-dimethylcyclopropyl)-4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-{1'-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
2-[1-(3-methylfuran-2-carbonyl)azetidin-3-yl]pyridine
2-benzyl-8-(prop-2-ene-1-sulfonyl)-2,8-diazaspiro[5.5]undecan-3-one
(4aR,8aR)-2-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-3-(piperazin-1-yl)propanamide
4-({5-[(2S)-piperidin-2-yl]-1,2,4-oxadiazol-3-yl}methyl)-1-propylpiperidine
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(4-methoxybenzenesulfonyl)pyrrolidin-3-yl]methanol
2,3-difluoro-4-methyl-N-[2-(pyrazin-2-yl)ethyl]benzamide
(1R,6S)-9-methyl-3-[(3-phenyl-1,2-oxazol-5-yl)methyl]-3,9-diazabicyclo[4.2.1]nonane
4-({1-[(2,3-dichlorophenyl)methyl]piperidin-2-yl}methyl)morpholine
2-[(2,5-difluorophenyl)methyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
2-(2-methoxy-4,6-dimethylpyridin-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
[(4aS,8aR)-6-(1-benzofuran-2-sulfonyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
3-benzyl-4-(2-fluoro-4-methylbenzoyl)piperazin-2-one
methyl 3-(2-chloro-6-fluorobenzamido)-6-{[(2-methoxy-2-oxoethyl)(methyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
9-[2-(methylsulfanyl)pyridine-3-carbonyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
methyl 4-{[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-[(pyridin-2-ylmethyl)amino]pyridine-3-carboxamide
2-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-4-carbonyl]-1,4-dihydroquinolin-4-one
4-(3-benzoylpiperidin-1-yl)-3-fluoropyridine
1,3-dimethyl-N-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-(2-ethoxyacetyl)-1-(4-methylphenyl)piperazin-2-one
4-[(2-methylprop-2-en-1-yl)oxy]-N-[1-(thian-4-yl)piperidin-4-yl]benzamide
(1R,5S,6S)-3-[(3,5-dichloro-2-hydroxyphenyl)methyl]-N-(2-hydroxyethyl)-N-methyl-3-azabicyclo[3.1.0]hexane-6-carboxamide
N-benzyl-4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidine-1-sulfonamide
4-{[1-(ethylcarbamoyl)piperidin-4-yl]amino}-N-(2-methoxyethyl)pyridine-2-carboxamide
dimethyl(2-{2-[1-(quinoxalin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
2-[2-({[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]acetic acid
1-[6-(1-hydroxyethyl)pyridin-2-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
8-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
4-[(2-methylpyrrolidin-1-yl)methyl]-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)benzamide
5-[7-(3-methoxypropyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]pyridine-2-carbonitrile
(1R,5R)-6-[(4-cyanophenyl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
9-(cyclopropylmethyl)-1-methyl-4-[2-(methylsulfanyl)pyrimidin-4-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}quinoline
4-{[8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile