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4-{2-[4-(5-ethylpyrimidin-2-yl)piperazin-1-yl]ethyl}morpholine
N-methyl-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)propanamide
2-(2,3-dimethylphenyl)-1H-1,3-benzodiazole-5-carbonitrile
1-(2-{4-[(3-fluorophenyl)methyl]-4-(hydroxymethyl)piperidine-1-carbonyl}phenyl)ethan-1-one
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3,5-dimethyl-1H-pyrazole-4-sulfonamide
2-[3-({[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)piperidin-1-yl]ethan-1-ol
{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
7-(cyclobutylmethyl)-2-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
8-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]-1-oxa-8-azaspiro[4.5]decane
9-methoxy-7-(4-methoxyphenyl)-4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
8-benzyl-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{2-[2-(3-fluorophenyl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydroquinolin-2-one
N-[4-({[1-(2-methyl-1,3-thiazol-4-yl)ethyl]carbamoyl}methyl)phenyl]butanamide
1-(6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-3-yl)ethan-1-one
(1r,4r)-4-{[2-(dimethylamino)-2-(2-methylphenyl)acetamido]methyl}cyclohexane-1-carboxylic acid
(1S,5R)-6-(cyclobutylmethyl)-3-(2-methyl-5-propylpyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(ethylamino)-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]pyrimidine-5-carboxamide
2-({1-[2-(3-methoxyphenyl)acetyl]azepan-3-yl}amino)pyridine-3-carboxamide
N-cyclopropyl-1-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
7-fluoro-3-methyl-2-(thiomorpholine-4-carbonyl)-1H-indole
6-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}pyridine-3-carboxamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-{2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}propan-1-one
N2,N2,5,6-tetramethyl-N4-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]pyrimidine-2,4-diamine
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-4-yl)-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
2-{4-[(2-methylpiperidin-1-yl)methyl]phenyl}-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
3-[1-(hydroxymethyl)-9-(2-methoxyethyl)-3,9-diazaspiro[5.5]undecan-3-yl]propanoic acid
(3-benzyl-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)methanol
2-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}acetamide
3-{4-azaspiro[2.5]octan-4-ylmethyl}-7-methyl-1,2-dihydroquinolin-2-one
4-(1H-pyrazol-3-yl)-N-(4-sulfamoylphenyl)piperidine-1-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(methylamino)pyridine-3-carboxamide
1-acetyl-N-[(3R,4S)-4-(propan-2-yl)-1-(pyrazin-2-yl)pyrrolidin-3-yl]piperidine-4-carboxamide
1-(4-methoxybenzoyl)-4-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperazine
N-methyl-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}-N-(propan-2-yl)acetamide
1-(2-{1-[(3-chloro-4-fluorophenyl)methyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
3-fluoro-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-5-methylimidazo[1,2-a]pyridine-2-carboxamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-[1-(pyridin-3-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1λ6-thiomorpholine-1,1-dione
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-methylpiperidine
ethyl 1-[1-(4-methylpyridin-2-yl)propan-2-yl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
1-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-N-(furan-2-ylmethyl)piperidine-4-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylpropanamide
1-{[6-(dimethylamino)pyridin-3-yl]methyl}-3-(2-methoxyethyl)piperidine-3-carboxylic acid
8-(3-methylbut-2-en-1-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(1-methylcyclopropyl)-1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)propan-1-one
N-(1,3-thiazol-2-yl)-2-({[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}amino)propanamide
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(2,5-dimethylfuran-3-carbonyl)piperidine-4-carboxylic acid
2-methyl-4-(2-methylphenyl)-1-(1H-pyrrole-2-carbonyl)piperazine
1-benzyl-N3-cyclopropyl-N5-[1-(6-methoxynaphthalen-2-yl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-propyl-3-(pyrrolidine-1-carbonyl)-N-[2-(thiophen-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine