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N-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-[(dimethylamino)methyl]pyrrolidin-3-ol
N-butyl-N-[(2-fluorophenyl)methyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
1-(2-ethoxyphenyl)-4-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperazine
2-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carbonitrile
3-methyl-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(propan-2-yloxy)phenyl]methyl}thiophene-2-carboxamide
2-(1,3-benzothiazol-2-yl)-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-{2-[methyl(phenyl)amino]propyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
(5S,9aS,9bS)-5-[5-methyl-2-(1H-pyrazol-1-yl)phenyl]-2-[(5-methylfuran-2-yl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-5-(oxolan-2-yl)thiophene-2-carboxamide
3-{2-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-oxoethyl}-1λ6-thiolane-1,1-dione
2-(4-methoxyphenyl)-N-{[1-(pyridin-4-ylmethyl)piperidin-3-yl]methyl}acetamide
N-(2,3-dihydro-1H-inden-2-yl)-3-ethyl-5-methyl-N-propyl-1,2-oxazole-4-carboxamide
2-[5-(2-chlorophenyl)-1,2,4-oxadiazol-3-yl]pyrazine
1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-3-ol
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-(5-methyl-1H-indazole-3-carbonyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
3-(2-oxo-2-{2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}ethyl)imidazolidine-2,4-dione
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-3-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
2-(dimethylamino)-1-(4-ethoxypiperidin-1-yl)-2-(3-methylphenyl)ethan-1-one
5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)-5-{1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
3-(4-methylphenyl)-5-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1,2,4-oxadiazole
8-(2-aminoacetyl)-2-[(3,4-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-(4-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}piperidin-1-yl)ethan-1-one
2-[1-(4-chlorophenyl)-5-oxo-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-[(5-methyl-1H-pyrazol-3-yl)methyl]acetamide
3-(2-fluorophenyl)-1-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
1-ethyl-N-(2-methoxyethyl)-N-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[1-(3-chlorophenyl)cyclopropyl]-2-fluoro-5-sulfamoylbenzamide
4-{[bis(prop-2-en-1-yl)amino]methyl}-N-(1-methyl-1H-1,2,4-triazol-3-yl)benzamide
5-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}-N-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
methyl 4-[(3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamido)methyl]benzoate
N-cyclopropyl-1-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)piperidine-3-carboxamide
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1-[4-(morpholine-4-carbonyl)phenyl]piperidin-4-amine
[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl](benzyl)(1,3-thiazol-2-ylmethyl)amine
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-(pyridin-4-yl)acetamide
1-[2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-1,2,3,6-tetrahydropyridine
1-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-3-(pyridin-4-yl)propan-1-one
{4-[(3-fluorophenyl)methyl]-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-4-yl}methanol
N-[4-chloro-3-({methyl[1-(1,2-oxazol-3-yl)ethyl]carbamoyl}amino)phenyl]-2-methoxyacetamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylbutanamide
2-methyl-6-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-3-yl}pyrimidin-4-ol
5-acetyl-N-(furan-2-ylmethyl)-N-(pyridin-4-ylmethyl)thiophene-3-carboxamide
3-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-1,6-dimethyl-1,2-dihydropyridin-2-one
6-[4-(1,3-benzoxazol-2-yl)piperazine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-methyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
N-[2-(3-methylpyridin-2-yl)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-[2-({2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)ethyl]pyridine-4-carboxamide
N-[(5-{[5-(hydroxymethyl)furan-2-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]cyclobutanecarboxamide
(3S,4S)-1-(2-amino-9H-purin-6-yl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
(4aR,7aS)-1-propyl-4-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S)-3-ethyl-4-[1-(pyridine-4-carbonyl)piperidine-4-carbonyl]morpholine