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N-methyl-N-[(3-methylthiophen-2-yl)methyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
2-(2,5-dimethylphenoxy)-N-(3-hydroxyadamantan-1-yl)propanamide
N-[2-(4-chlorophenyl)ethyl]-3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
2-(3,3-diphenylpiperidine-1-carbonyl)-5-methoxy-4H-pyran-4-one
3-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-1,3-oxazolidin-2-one
6-(2-fluoro-4-methoxyphenyl)-N-(2-hydroxypropyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-(2-{2-[2-(2-methylphenyl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
{3-[(2-methylphenyl)methyl]-1-(oxan-4-yl)piperidin-3-yl}methanol
(1R,2S)-1-{2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}-2,3-dihydro-1H-inden-2-ol
3-{5-oxo-3-[1-(1H-pyrazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-4-yl}propanoic acid
1-[2-(4-chlorophenyl)ethyl]-N-[(5-fluoro-2-methylphenyl)methyl]-6-oxopiperidine-3-carboxamide
N-{1-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-4-yl]-2-phenylethyl}-N-methylthiophene-2-carboxamide
2-methyl-3-{3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1,8-naphthyridine
N-[1-(cyclohexylmethyl)-1H-pyrazol-5-yl]-2-{1H-pyrazolo[3,4-b]pyridin-1-yl}acetamide
4-hydroxy-2-methyl-N-[3-(propan-2-yloxy)propyl]pyrimidine-5-carboxamide
N4-(furan-2-ylmethyl)-N1-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}piperidine-1,4-dicarboxamide
1-(cyclohex-3-en-1-ylmethyl)-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
3-(azepan-1-ylmethyl)-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
(4aR,8aS)-6-(1-methylpiperidin-4-yl)-1-(pyridin-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
N-[(3S,4R)-4-(4-methylphenyl)-1-(4-methylpyrimidine-5-carbonyl)pyrrolidin-3-yl]cyclopropanecarboxamide
2-{4-[5-(1H-1,2,4-triazol-1-ylmethyl)-1,2,4-oxadiazol-3-yl]phenyl}ethan-1-ol
4-hydroxy-N-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
1-[benzyl(methyl)amino]-3-[4-({[2-(pyrrolidin-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
7-[2-(4-fluorophenoxy)acetyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-ethyl-3-(piperidine-1-carbonyl)-N-[3-(propan-2-yloxy)propyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
(1S,6R)-9-[5-(piperidine-1-carbonyl)pyridin-2-yl]-3,9-diazabicyclo[4.2.1]nonan-4-one
1-[4-({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]amino}methyl)thiophen-2-yl]ethan-1-one
methyl 1-(2-methylpropyl)-3-(2-phenylacetamido)-5-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
N-{[6-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,3-thiazole-5-carboxamide
2-{4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
3-(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(furan-2-yl)ethyl]propanamide
[(2,5-dimethoxyphenyl)methyl](methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
(2S,4S)-N-ethyl-4-(4-{2-[(2-methylphenyl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxamide
1-{2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-3-phenoxypropan-1-one
3-({2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-1,2-dihydroquinoxalin-2-one
4-phenyl-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
4-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-(prop-2-en-1-yl)pyrrolidin-2-one
2-methyl-4-{3-[4-(oxan-4-yl)piperazine-1-carbonyl]phenyl}butan-2-ol
4-(1H-imidazol-2-yl)-1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-1,2,3-triazole
2-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}-1,2-oxazinane
2-cyclopentyl-9-(1H-pyrazole-4-sulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-butyl-N-[(5-methylthiophen-2-yl)methyl]-2-(4-oxo-1,4-dihydroquinolin-1-yl)acetamide
6,7-dimethyl-4-{[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl}-2H-chromen-2-one
5-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidine-1-carbonyl]pyridine-2-carbonitrile
2-{2-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-ylmethyl]phenoxy}-1-(piperidin-1-yl)ethan-1-one
4-(5-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)pyridine
(1S,5R)-6-(pyridin-2-ylmethyl)-3-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
6-chloro-N,N-dimethyl-3-[(3-phenoxyazetidin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide