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1-cycloheptyl-N-[(4-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
N-methyl-2-(phenylamino)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide
5-[2-(methylsulfanyl)phenyl]-1-propyl-1H-1,2,4-triazole
1-{2-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]-6-methoxyphenyl}ethan-1-one
1-({2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl}methyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(3-chloro-4-propoxyphenyl)-3-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]urea
5-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrazine-2-carboxylic acid
(2S,4R)-4-amino-N,N-diethyl-1-[(4-methyl-1H-imidazol-5-yl)methyl]pyrrolidine-2-carboxamide
5-[(E)-2-phenylethenyl]pyridine-3-carboxamide
3-methyl-5-[(2-phenyl-1H-imidazol-1-yl)methyl]-1H-1,2,4-triazole
3-{[(furan-3-ylmethyl)(methyl)amino]methyl}-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
(1-{[1-(2,6-dimethylquinoline-4-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanamine
3-[(1S,4S)-3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
methyl 4-({[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)benzoate
2-{[1-(4-cyclopentyl-3-oxopiperazin-1-yl)-1-oxopropan-2-yl]sulfanyl}-6-methyl-3,4-dihydropyrimidin-4-one
(1R,2R,4R)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
4-chloro-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-methyl-1H-pyrazole-3-carboxamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-5-chloro-2,3-dihydro-1H-indole-2-carboxamide
3-[(3S,4R)-1-benzyl-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-1-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]propan-1-one
1-{imidazo[1,2-a]pyrimidin-6-ylmethyl}-4-[(3-methylphenyl)methyl]piperazine
(3S)-1-[1-(4-methoxyphenyl)-5-phenyl-1H-pyrazole-3-carbonyl]pyrrolidin-3-amine
1-ethyl-4-{[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}pyrrolidin-2-one
N-[(2,5-dimethoxyphenyl)methyl]-5-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)pentanamide
1-cyclopropyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-5-oxopyrrolidine-3-carboxamide
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(4-chloro-3-methyl-1H-pyrazol-1-yl)ethan-1-one
2-(2-methylphenyl)-5-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)pyrimidine
N-methyl-2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}butanamide
(1R,5S,6S)-6-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]-3-azabicyclo[3.1.0]hexane
N'-[3-(pyridin-4-yl)propyl]-N-(2,4,6-trimethylphenyl)butanediamide
4-(1H-imidazol-1-yl)-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidine-4-carboxylic acid
1-cycloheptyl-N-methyl-N-(oxan-4-yl)-6-oxopiperidine-3-carboxamide
4-{[1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)piperidin-2-yl]methyl}morpholine
3-fluoro-2-{3-[1-(pyridin-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridine
1-(4-cyclohexylphenyl)-3-(1,1-dioxo-1λ6-thiolan-3-yl)-3-ethylurea
4-[2-(furan-2-ylmethoxy)phenyl]-4H-1,2,4-triazole
[(2R)-1-{[2-(3,4-dimethoxyphenyl)-7-methylquinolin-3-yl]methyl}pyrrolidin-2-yl]methanol
(2S,4R)-4-(6-methyl-4-oxo-4H-pyran-2-amido)-1-[(2E)-2-methylbut-2-en-1-yl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-[5-(4H-1,2,4-triazol-4-yl)pentyl]morpholine
N-cycloheptyl-2-[7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]acetamide
1-(2-methoxyethyl)-4-[4-(5,6,7,8-tetrahydronaphthalen-2-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
N-[(3S,4R)-1-(5-hydroxypyrazine-2-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}-2-(methylsulfanyl)pyridine-3-carboxamide
3-[(2R,3R,6R)-5-[(3-fluoropyridin-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
2-(pyridin-3-ylmethyl)-8-(pyrimidin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
4-[2-(3-methoxyphenoxy)ethyl]-1,3λ6,4-oxathiazinane-3,3-dione
4-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)sulfonyl]piperazine-2-carboxylic acid
2-{4-[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyridine-3-carboxamide
1-[(2-fluorophenyl)methyl]-4-[4-(3-methoxyphenyl)-5-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl]piperidine
N-(2-{3-hexyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)-2-methylpropanamide
{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}[(5-fluoro-1H-indol-2-yl)methyl]methylamine