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4-(4-fluoro-2-methylphenoxy)-1-(oxolane-3-carbonyl)piperidine-4-carboxylic acid
5-ethyl-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-[2-(1H-pyrazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(5-{4-[(propan-2-yl)amino]pyrimidin-2-yl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]cyclobutanecarboxamide
1-[(4-methylphenyl)methyl]-3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
2-acetyl-8-(pyrrolidine-1-sulfonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-methoxy-2-[(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]pyridin-4-ol
N-(1-carbamoylcyclopentyl)-6-fluoro-4-hydroxyquinoline-3-carboxamide
8-[(furan-2-ylmethyl)carbamoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(4aS,8aR)-6-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2-methyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrido[2,3-d]pyrimidin-4-amine
3-(2-{8-[2-(1H-imidazol-4-yl)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-oxoethyl)imidazolidine-2,4-dione
N-(1,2-diethyl-1H-1,3-benzodiazol-5-yl)-4-(pyrimidin-2-yl)piperazine-1-carboxamide
2-(2-chlorophenyl)-3-methyl-N-(oxan-4-yl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-(1H-1,3-benzodiazol-1-yl)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]acetamide
1-[(4aR,8aS)-6-benzyl-decahydro-1,6-naphthyridin-1-yl]-2-(1,3-thiazol-4-yl)ethan-1-one
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-[(3-methoxyphenyl)sulfanyl]ethan-1-one
3-{1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-4,6-dimethyl-2-oxo-2H-pyran-5-carboxamide
(3S,4S)-1-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-(dimethylamino)pyrrolidin-3-ol
N-(3-cyano-4-ethoxyphenyl)-3-(3-methoxypropyl)piperidine-1-carboxamide
2-(4-fluorophenyl)-4-[5-(morpholine-4-carbonyl)pyridin-2-yl]morpholine
(3aS,6aS)-2-(2-hydroxyethyl)-5-[(6-methoxynaphthalen-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[3-(2-methylphenyl)-3-phenylpropanoyl]piperazin-2-one
1-(1-{4-[(pyridin-4-ylmethyl)amino]benzoyl}piperidin-4-yl)pyrrolidin-2-one
5-methyl-4-[(2-methylpyridin-3-yl)oxy]-6-[4-(piperazin-1-yl)piperidin-1-yl]pyrimidine
8-[1-(furan-2-ylmethyl)piperidin-4-yl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-chloro-2-({4-[1-(propan-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-1-yl}methyl)-1H-1,3-benzodiazole
7-(3-chlorophenyl)-4-[(4,6-dimethylpyrimidin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-{[(1-methyl-1H-imidazol-2-yl)methyl]({[4-(methylsulfanyl)phenyl]methyl})amino}ethan-1-ol
N-methyl-5-(phenoxymethyl)-N-(quinolin-2-ylmethyl)-1H-pyrazole-3-carboxamide
8-[2-(3-acetyl-1H-indol-1-yl)butanoyl]-2,8-diazaspiro[4.5]decan-3-one
8-[(3-hydroxyphenyl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-(1H-pyrazol-5-yl)piperidine
8-[2-(benzyloxy)acetyl]-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(1H-imidazol-1-yl)ethyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-4-(4H-1,2,4-triazol-4-yl)benzamide
N-[2-(1H-imidazol-4-yl)ethyl]-6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
(1S,5R)-3-{9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-sulfamoylbenzamide
1-[1-(oxan-4-yl)piperidine-4-carbonyl]azepan-3-amine
4-[(3-methylphenyl)methyl]-1-(2-phenoxyacetyl)-1,4-diazepan-5-one
(4aS,8aR)-6-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
4-(2-hydroxy-5-methoxyphenyl)-8-methyl-7-(pyrrolidin-1-yl)-1,2,3,4-tetrahydroquinolin-2-one
3-[2-(3,4-difluorophenyl)ethyl]-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-2-carboxamide
5-{[methyl({[3-(2-{4-[4-(trifluoromethyl)benzoyl]piperazin-1-yl}ethoxy)phenyl]methyl})amino]methyl}pyrrolidin-2-one
2-({[(3R,4R)-1-(7-chloro-1-methyl-1H-indole-2-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol