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5-(2-{2-ethyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-butyl-4-(2-ethylpyrimidine-5-carbonyl)-1-(3-methylphenyl)piperazin-2-one
2-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)phenoxy]acetamide
1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(2-methoxyethyl)piperidine
4-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenol
3-fluoro-4-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
N-{2-[4-(dimethylamino)phenyl]ethyl}-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
3,5-dimethyl-N-[1-(methylcarbamoyl)cyclohexyl]-1H-indole-2-carboxamide
5-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one
2-chloro-N-{1-[1-(3-cyclopentylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
2-methyl-4-phenyl-9-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-2,9-diazaspiro[5.5]undecane
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-8-[5-(trifluoromethyl)pyridin-2-yl]-1,8-diazaspiro[4.5]decane
1-{3-[(1,4-dithiepan-6-yl)amino]azepan-1-yl}pentan-1-one
1-(4-cyclopropanecarbonylphenyl)-2-propyl-1H-imidazole
(3R,5R)-N-[2-(dimethylamino)ethyl]-1-(naphthalen-2-ylmethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
N-(1-methylpiperidin-3-yl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[(1,2-oxazol-3-ylmethyl)amino]methyl}piperidin-2-one
methyl 5-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
5-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N,1,3-trimethyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(4-{[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}phenyl)imidazolidin-2-one
(1H-imidazol-2-ylmethyl)(methyl){[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amine
4-(cyclohex-3-en-1-yl)-1-[(2,6-difluoro-3-methylphenyl)methyl]-1H-1,2,3-triazole
3-[({1-[2-(1H-pyrazol-1-yl)benzoyl]piperidin-3-yl}oxy)methyl]pyridine
4-(2-methylphenoxy)-1-(pyridin-3-ylmethyl)piperidine-4-carboxylic acid
N-[2-(4-methoxyphenyl)ethyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
9-[(4-fluorophenyl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-butyl-4-(2-ethoxypyridine-3-carbonyl)-1-methylpiperazin-2-one
N-{1-[(2-chlorophenyl)methyl]-3-methyl-1H-pyrazol-5-yl}-1H-1,3-benzodiazole-5-carboxamide
N-ethyl-3-(morpholine-4-carbonyl)-1-propyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2-ethoxy-5-{[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]methyl}phenyl)methanol
N-[(3-methylphenyl)methyl]-2-oxo-N-(propan-2-yl)-2-(pyrrolidin-1-yl)acetamide
2-(2-propyl-1H-1,3-benzodiazol-1-yl)-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}propanamide
diethyl({3-[(2S)-2,4,5,5-tetramethylpiperazine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
4-{6-[(3-methoxyphenyl)methoxy]-3-oxo-4-(2-phenylethyl)-1,4-diazepane-1-carbonyl}-2-methyl-1,2-dihydrophthalazin-1-one
6-methyl-5-(2-oxo-2-{2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-methyl-6-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1,3-benzoxazole
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1-(morpholin-4-yl)cyclohexane-1-carboxamide
N-{[4-(oxolan-3-yloxy)phenyl]methyl}-3-(2-oxopyrrolidin-1-yl)-N-(pyridin-2-ylmethyl)benzamide
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]benzamide
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-(1H-pyrazol-3-yl)piperidine
1-(2-ethyl-6-methylphenyl)-4-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
N-[2-(azepan-1-yl)ethyl]-N-methyl-4-(pyridin-2-yl)pyrimidin-2-amine
1-({1-[3-(1H-imidazol-1-yl)butanoyl]piperidin-4-yl}methyl)pyrrolidin-2-one
1-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(pyridin-3-yl)propan-1-one
N-[2-(1H-indol-3-yl)ethyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
1-({1-[1-(phenylamino)cyclopentanecarbonyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
(2H-1,3-benzodioxol-4-ylmethyl)[(2-fluorophenyl)methyl](2-methoxyethyl)amine
{1-[4-(5,6-dimethylpyrimidin-4-yl)phenyl]ethyl}dimethylamine