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6-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]pyridin-2-ol
2-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-(4-hydroxyphenyl)acetic acid
8-(5-chloropyridin-2-yl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
[(3aS,6aS)-2-(3-phenyl-1H-pyrazole-4-carbonyl)-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
3-(3-chlorobenzoyl)-1-(propane-1-sulfonyl)piperidine
1-(3-{[3-(4-cyclopentylpiperazine-1-carbonyl)-1H-pyrazol-5-yl]methoxy}phenyl)ethan-1-one
1-(cyclopropylmethyl)-5-({2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}amino)azepan-2-one
1-(1-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}azetidin-3-yl)-3,5-dimethyl-1H-pyrazole
2,5-dimethoxy-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]benzamide
6-{[(2-aminopyridin-3-yl)methyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
ethyl 4-[4-hydroxy-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-amido]piperidine-1-carboxylate
3-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
(3S,9aR)-3-(cyclohexylmethyl)-8-[4-(trifluoromethoxy)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(2R,6R)-4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(3aS,6aS)-2-(3-chloropyridin-2-yl)-5-(ethanesulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1'-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-[(2R,3R,6R)-5-[(1-methyl-1H-imidazol-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
ethyl 3-[(4-fluorophenyl)methyl]-1-(3-methoxybenzoyl)piperidine-3-carboxylate
3-(1-cycloheptylpiperidin-3-yl)-1-phenylurea
3-chloro-6-{4-[(6-phenoxypyridin-3-yl)methyl]piperazin-1-yl}pyridazine
4-{[4-(1,3-dihydroxypropan-2-yl)-6-hydroxy-1,4-diazepan-1-yl]methyl}benzamide
4-(5-methyl-1,2,4-oxadiazol-3-yl)-1-(oxolan-3-ylmethyl)piperidine
N-[(2S)-4-(methylsulfanyl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-1-oxobutan-2-yl]acetamide
2-(5-acetylthiophen-3-yl)-N-[2-oxo-2-(piperazin-1-yl)ethyl]acetamide
4-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-4-oxobutanamide
4-[(5-acetylthiophen-3-yl)methyl]-1-[(2-fluorophenyl)methyl]piperazin-2-one
N-{1-[4-(4-chlorophenyl)butanoyl]piperidin-4-yl}methanesulfonamide
5-(4-fluorophenyl)-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-ethyl-4-{[1-(4-fluoro-3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-3-methyl-1H-pyrazole
5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1,2-oxazole-3-carboxamide
N-{5-[2-(3-acetylphenyl)-1H-imidazol-1-yl]-2-fluorophenyl}-2-methylpropanamide
{4-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]morpholin-2-yl}methanamine
2-amino-3-ethyl-N-[(4-fluorophenyl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]-2-(pyrrolidin-1-yl)ethan-1-one
1-(2,6-dimethylpyridin-4-yl)-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperazine
2-(2H-1,2,3-benzotriazol-2-yl)-N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}acetamide
3-fluoro-4-methoxy-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}benzamide
8-fluoro-2-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]quinoline
{3-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]phenyl}methanamine
ethyl 1-{1-benzyl-4-oxo-5-[(propan-2-yl)carbamoyl]-1,4-dihydropyridine-3-carbonyl}piperidine-2-carboxylate
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)(methyl)(quinolin-2-ylmethyl)amine
(1S,4S)-5-[(2R)-2-hydroxypropanoyl]-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
N-[(6-fluoroquinolin-2-yl)methyl]-N-(3-methoxypropyl)-1-methylpiperidin-4-amine
2-(2-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(1-methyl-1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclopentyl-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(prop-2-en-1-yl)acetamide
[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl)({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)amine
1-(4-{4-azaspiro[2.5]octan-4-ylmethyl}-2-methoxyphenoxy)-3-(morpholin-4-yl)propan-2-ol
(2S)-2-amino-3-(1H-imidazol-4-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)propanamide
2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one