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2-{1-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-1-oxobutan-2-yl}-2,3-dihydro-1H-isoindol-1-one
methyl 5-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
4-[2-(2-{[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenoxy)ethyl]morpholine
2-[1-(oxan-4-ylmethyl)-1H-imidazol-2-yl]-1-propyl-1H-imidazole
N-[2-(dimethylsulfamoyl)ethyl]-2,3-dimethyl-1H-indole-5-carboxamide
9-(2-methoxyethyl)-1-methyl-4-(5-methylthiophene-2-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
4-[4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1-methylpiperazin-2-one
3-chloro-4-{[1-(2-hydroxyacetyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]acetamide
methyl 4-{[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}benzoate
8-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{[(3-tert-butyl-1H-pyrazol-5-yl)methyl]amino}pyrimidine-5-carboxylic acid
N-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
[(1,5-dimethyl-1H-indol-2-yl)methyl][(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]methylamine
3-(4-ethyl-1H-pyrazol-5-yl)-1-[3-(1H-pyrazol-4-yl)benzoyl]piperidine
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-(propan-2-yl)-2-(5,6,7,8-tetrahydronaphthalen-2-yloxy)butanamide
1-[2-(dimethylamino)-2-(furan-2-yl)ethyl]-3-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
N-[(3-fluoro-4-methoxyphenyl)methyl]-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
8-fluoro-N-(2-hydroxyethyl)-4-oxo-N-(thiophen-2-ylmethyl)-1,4-dihydroquinoline-3-carboxamide
(2R,6R)-4-[(5-acetylthiophen-3-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4,4,4-trifluoro-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]butanamide
1-(morpholin-4-yl)-3-[5-(pyridin-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propan-1-one
2-[2-(isoquinolin-5-yl)phenoxy]propanamide
2-(4-{[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}phenoxy)propanoic acid
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
1-[2-(dimethylamino)-4-{[(4-ethyl-1,3-thiazol-2-yl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-(3-ethoxypropyl)-4-{[2-(1H-indol-3-yl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
(4aS,8aR)-6-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-(3-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}-2,5-dimethyl-1H-pyrrol-1-yl)acetamide
5-methyl-1-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-5-phenylpiperidin-2-one
N,N,4-trimethyl-3-({[2-(1,3-thiazol-4-yl)ethyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-cyclopentyl-5-{4-hydroxy-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1-benzofuran-2-carboxamide
5-cyano-N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
(2S,4R)-4-amino-N,N-diethyl-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}pyrrolidine-2-carboxamide
6-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[(1R,5S,6R)-6-({methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)-3-azabicyclo[3.1.0]hexane-3-carbonyl]benzonitrile
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-[3-(1H-imidazol-1-yl)pyrrolidin-1-yl]ethan-1-one
1-[(4-chlorophenyl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
1-methyl-3-(2-methylpropyl)-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
5-propyl-1'-(1H-pyrrole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N,4-dimethyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
1-(2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
3-tert-butyl-1-({1-[(3-methylphenyl)methyl]piperidin-4-yl}methyl)urea
N-methyl-2-(1-oxo-1,2-dihydroisoquinolin-2-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
3-{imidazo[1,2-a]pyridin-2-yl}-1-[2-(3-methoxyphenyl)azetidin-1-yl]propan-1-one
2-[4-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-[(4-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
N-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
3-[4-(oxolan-2-ylmethyl)piperazin-1-yl]-N-[4-(propan-2-yl)phenyl]propanamide
1-[(2-methylphenyl)methyl]-4-(3,3,3-trifluoro-2-methylpropyl)piperazine