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7-{3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]propanoyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(1-cyclopentylpiperidin-4-yl)methyl]({[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
N-[3-(tert-butylcarbamoyl)-2-methylphenyl]-1,2,3-thiadiazole-4-carboxamide
3-[5-(1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidin-3-yl)-1,2,4-oxadiazol-3-yl]pyridine
N-{[1-(5-ethyl-1,2,4-oxadiazol-3-yl)piperidin-3-yl]methyl}-4-methoxybenzene-1-sulfonamide
N-{[7-fluoro-5-(3-fluoro-4-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-imidazol-1-yl)propan-1-one
2-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)-5-methylpyrimidin-4-amine
methyl({[2-(piperidin-1-yl)pyrimidin-5-yl]methyl})[1-(pyridin-2-yl)ethyl]amine
4-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}pyrimidine
2-methoxy-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
{2-oxo-2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}urea
2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1,3-oxazole
9-(4-methylquinolin-2-yl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-N-(1-{1-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
1-(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazin-1-yl)-3-(1-methyl-1H-pyrazol-5-yl)propan-1-one
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-cyclopentyl-2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propanamide
4-(4-fluorophenyl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-oxobutanamide
[2-ethoxy-5-({[(3R)-oxolan-3-yl]amino}methyl)phenyl]methyl acetate
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(2-hydroxybutyl)-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
9-[(1S,3R)-3-aminocyclopentanecarbonyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(4aS,7aR)-1-[(3,5-dimethylphenyl)methyl]-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[2-(1H-imidazol-4-yl)ethyl]-8-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-methyl-4-[4-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenyl]butan-2-ol
2-{2-[5-(1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-7-methyl-1H-1,3-benzodiazole
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrrolidine-3-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(pyridine-2-carbonyl)piperidin-3-ol
3-(3-methoxypyrrolidine-1-carbonyl)-N-[2-(1H-pyrazol-1-yl)ethyl]benzene-1-sulfonamide
N-[(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)methyl]cyclohexanecarboxamide
3-(2-methoxyethyl)-5-(4H-1,2,4-triazol-4-ylmethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
3-(2-amino-1,3-thiazol-4-yl)-1-[2-(3-methoxyphenyl)pyrrolidin-1-yl]propan-1-one
9-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-1,4,9-triazaspiro[5.5]undecan-5-one
1-benzyl-6-methoxy-4-[1-(2-phenylethyl)piperidin-4-yl]-1,4-diazepan-2-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-4-hydroxy-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
N-methyl-5-{[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]methyl}furan-2-carboxamide
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
(3S,4R)-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-(thiophen-2-yl)ethane-1,2-dione
3-{1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]piperidin-3-yl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(5-methyl-1,3,4-oxadiazol-2-yl)-1-(pyrazin-2-yl)piperidin-3-amine
4-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}-1-(2-methylpropyl)piperidine
3-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-1-(3-hydroxy-3-phenylpropyl)-1-methylurea
N-[4-({[(5-fluoro-1H-indol-2-yl)methyl](methyl)amino}methyl)phenyl]acetamide
ethyl 1-(2-acetamidoacetyl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
5-(2,2-dimethylpropanoyl)-N-(3-phenylpropyl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-8-methoxy-3,4-dihydro-2H-1-benzopyran