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2-(4-acetylphenoxy)-N-{[5-(3,6-dimethylpyrazin-2-yl)-7-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N,N-dimethyl-4-[({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1,3-thiazol-2-amine
ethyl 1-[(5-chloro-2-methylphenyl)carbamoyl]-4-[(4-chlorophenyl)methyl]piperidine-4-carboxylate
N-(1H-1,2,3-benzotriazol-5-yl)-2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carboxamide
N3-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-N5-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(4-oxo-3,4-dihydroquinazolin-3-yl)propanamide
2-(3-fluorophenoxymethyl)-4-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1,3-oxazole
N-[(1R,2S)-2-phenylcyclopropyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[2-(1-methylpiperidin-2-yl)ethyl]-6-[(1-methylpiperidin-4-yl)amino]pyridine-3-carboxamide
1-acetyl-N-[4-(1,3-benzoxazol-2-yl)phenyl]pyrrolidine-2-carboxamide
(1R,7S)-3-(3,4-dimethylphenyl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2,3-dimethyl-7-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]-1H-indole
[(4-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}-1,3-thiazol-2-yl)methyl]dimethylamine
1-(2-{[(1,3-benzothiazol-2-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
N-{1-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]propan-2-yl}acetamide
5-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidine-1-carbonyl]-4-ethyl-1,3-thiazol-2-amine
N-(furan-2-ylmethyl)-N-methyl-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2R,3R)-3-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-{[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]amino}-N-cyclohexylpropanamide
(3E)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}hex-3-enamide
1-(2,5-dimethoxyphenyl)-2-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethan-1-ol
2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}[2-(dimethylamino)ethyl]amino)ethan-1-ol
methyl[1-(pyridin-3-yl)propyl](thiophen-3-ylmethyl)amine
1-methyl-4-(3-methylthiophen-2-yl)-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[2-(3-phenylpiperidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
4-[1-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-4-yl)ethyl]morpholine
[(4-chloro-1-methyl-1H-indazol-3-yl)methyl](methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-(3-hydroxyphenyl)ethan-1-one
1-ethyl-3-[(3S,4S)-3-[ethyl(methyl)amino]-4-hydroxypyrrolidine-1-carbonyl]-7-methyl-1,4-dihydro-1,8-naphthyridin-4-one
N-{2-[1-(4-chloro-2-hydroxybenzoyl)piperidin-2-yl]ethyl}acetamide
3-[2-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-oxoethyl]-5,5-dimethylimidazolidine-2,4-dione
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-3-(3-methoxyphenyl)propanamide
3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-pyrrole-3-carbonyl)piperidine
3-(2-fluorophenyl)-3-phenyl-N-[2-(pyridin-4-yl)ethyl]propanamide
1-benzyl-N,N-dimethyl-5-({[1-(piperidin-1-yl)cyclohexyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[2-(piperidin-1-ylmethyl)phenoxy]-6-(pyrrolidine-1-carbonyl)pyrazine
2-[5-(1-methylazepan-2-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]acetic acid
N-benzyl[(2-amino-6-methyl-1,3-benzothiazol-4-yl)amino]sulfonamide
3-[(3R,4S)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
(2R,6S)-1-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)-2,6-dimethylpiperidine
1-{1-[2-amino-6-(2-methylpropyl)pyrimidine-4-carbonyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-methyl-N-(2-methylpropyl)-1,3-oxazole-4-carboxamide
ethyl 1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-4-(2-phenylethyl)piperidine-4-carboxylate
2-{2-amino-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-tert-butylbenzene-1-sulfonamide
methyl 4-({2-[2-(dimethylamino)ethyl]morpholine-4-carbonyl}amino)benzoate
11-[ethyl(2-methylprop-2-en-1-yl)amino]-4-[3-(propan-2-yloxy)propyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-methyl-2-{4-[6-(thiomorpholin-4-yl)pyridazin-3-yl]phenyl}propanenitrile
N,N-bis(2-methoxyethyl)-2-[(3-methoxyphenyl)amino]butanamide
{[3,5-dichloro-4-(prop-2-en-1-yloxy)phenyl]methyl}[1-(1H-1,2,4-triazol-5-yl)ethyl]amine
4-{[1-(4-fluoro-3-methylbenzoyl)piperidin-2-yl]methyl}morpholine