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1-benzyl-4-[3-(hydroxymethyl)quinolin-2-yl]-1,4-diazepan-6-ol
N-[(4-fluorophenyl)methyl]-3-[1-(thiophene-3-carbonyl)piperidin-4-yl]propanamide
4-methyl-2-(propan-2-yl)-N-{3-[(pyridin-3-yl)amino]propyl}-1,3-thiazole-5-carboxamide
1-({1-[(2-phenylethyl)carbamoyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-(1H-pyrazol-1-yl)acetamide
2-[(3S,4R)-3-[(dimethylcarbamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-N-(2-phenylethyl)acetamide
7-{5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carbonyl}-2-oxa-7-azaspiro[4.5]decane
1-(diethylamino)-3-(2-methoxy-5-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
N-(2,4,6-trimethylpyridin-3-yl)thiomorpholine-4-carboxamide
2-({7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}sulfanyl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]acetamide
2-{4-[1-(3-fluoro-4-methylbenzoyl)piperidin-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}ethan-1-ol
2-(3-methoxypropyl)-9-(pyridine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N,N,4-trimethyl-3-({[(methylcarbamoyl)methyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-3-(4-methoxyphenoxymethyl)piperidine
N,1,3-trimethyl-2,6-dioxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-(4-chlorophenyl)-5-({4-[2-(methylsulfanyl)ethyl]piperazin-1-yl}methyl)pyrimidine
2-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-5-propyl-1,3,4-oxadiazole
5-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]-1H-1,3-benzodiazole
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)acetamide
N-(cyclohexylmethyl)-N-ethyl-2-methanesulfonylacetamide
2-[1,4-bis(cyclohexylmethyl)piperazin-2-yl]ethan-1-ol
N-({8-benzyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-[(5Z)-2,4-dioxo-1,3-thiazolidin-5-ylidene]acetamide
2-{[2-(1,3-thiazol-2-yl)piperidin-1-yl]methyl}benzonitrile
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
1-(4-fluoro-2-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}phenyl)-1H-pyrazole
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
2-(dimethylamino)-2-(4-methylphenyl)-N-(1,2-oxazol-3-ylmethyl)acetamide
1-methyl-N-(2,2,2-trifluoroethyl)-1H-indole-6-carboxamide
7-methyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-4-oxo-4H-chromene-2-carboxamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(1,3-thiazol-5-yl)acetamide
5-{[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]sulfanyl}-1H-1,2,3-triazole
N-methyl-4-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
N-{[4-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1-[(4-methylphenyl)methyl]-5-oxopyrrolidine-3-carboxamide
N-{[5-(pyridin-2-yl)thiophen-2-yl]methyl}-2-(pyrrolidin-3-yl)benzamide
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]methylamine
2-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-3,5,7-trimethyl-1H-indole
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}benzamide
2-(methylsulfanyl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-(cyclohex-1-ene-1-carbonyl)-4-[(2-fluorophenyl)methyl]-1,4-diazepan-5-one
2-ethoxy-5-{2-[(oxolan-3-ylmethyl)amino]pyrimidin-4-yl}benzoic acid
4-({[(1S)-1-carbamoyl-2-phenylethyl]amino}methyl)-2,6-dimethylphenyl acetate
1-(1-methyl-1H-pyrazole-3-carbonyl)-4-(piperidine-1-carbonyl)piperidine
4-ethyl-3-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(1H-imidazol-2-ylmethyl)({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amine
N-[(3R,4R)-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
dimethyl[2-(1-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}piperidin-2-yl)ethyl]amine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-ol
3-({5-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-4-phenyl-1H-imidazol-1-yl}methyl)-5-methyl-4H-1,2,4-triazole
N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-6-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide