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5-hydroxy-1,2-dimethyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1H-indole-3-carboxamide
methyl 2-[(butan-2-yl)sulfamoyl]-6-{2-[4-(methylsulfanyl)phenyl]acetyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-[(3-methoxypropyl)amino]-5-methyl-N-(thiophen-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
{[4-ethyl-5-(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
(1R,3s,6r,8S)-4-[6-(piperidin-4-yl)pyrimidin-4-yl]-4-azatricyclo[4.3.1.13,8]undecane
2-amino-7-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-methylpiperidine-4-carbonitrile
3-(3-methyl-1H-1,2,4-triazol-5-yl)-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-1-carboxamide
N-methyl-3-(1H-pyrazol-1-ylmethyl)-N-(quinolin-4-ylmethyl)benzamide
1-methyl-4-[5-methyl-6-(4-methylpiperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-yl]piperazine
4-(2-hydroxy-5-methoxyphenyl)-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(2-{[4-(4-methylphenyl)-5-(pyridin-3-yl)pyrimidin-2-yl]amino}ethyl)piperidin-3-ol
N-[2-(azepan-1-yl)ethyl]-4-chloro-N-methyl-1H-indole-2-carboxamide
7-[(2,3-dimethoxyphenyl)methyl]-2-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-2,7-diazaspiro[4.5]decane
2-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}phenol
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
{4-benzyl-1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}methanol
2-{[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]methyl}benzonitrile
4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
2-{[5-(carboxymethyl)pyrimidin-4-yl]amino}-4-(methylsulfanyl)butanoic acid
3-{[(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)amino]methyl}pyrrolidin-3-ol
2-methyl-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl 6-{[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidin-1-yl]methyl}pyridine-2-carboxylate
2-{[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl](methyl)amino}-N,N-dimethylpropanamide
1-(3-methoxyphenyl)-4-(3-methyl-1H-pyrazole-5-carbonyl)piperazin-2-one
2-(3-methyl-1H-1,2,4-triazol-5-yl)-N-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)pyrrolidine-1-carboxamide
3-({3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}methyl)-6-methyl-4H-chromen-4-one
3-(ethylsulfanyl)-1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamide
(3S,4R)-4-(2-methoxyphenyl)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]pyrrolidine-3-carboxylic acid
2,6-dimethoxy-4-(1-methyl-1H-1,3-benzodiazol-2-yl)phenol
2-methoxy-1-[1'-(thiophene-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-4-(1H-pyrazol-1-yl)butan-1-one
2-amino-7-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
6-(2-methylquinolin-5-yl)-2-(morpholin-4-yl)pyrimidin-4-amine
8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-{[3-(methylsulfanyl)phenyl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
1-(4-fluoro-3-methoxyphenyl)-3-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}urea
methyl 6-[(4-methoxy-2,5-dimethylphenyl)methyl]-2-[(propan-2-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-{[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
N-cyclopropyl-2-[4-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)piperidin-1-yl]acetamide
(2S,4R)-4-{[(2,5-dimethylphenyl)methyl]amino}-N-methyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-[(1S)-1-phenylethyl]-3-[(propan-2-yl)sulfamoyl]-5-[(thiophen-2-ylmethyl)amino]benzamide
2-(3-methoxypropanoyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-ethyl-N-propylpropanamide
ethyl 2-[4-(4-fluorobenzenesulfonyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl]acetate
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4,6-dimethoxypyrimidine
2-amino-4-(5-cyano-1-methyl-1H-pyrrol-3-yl)-6-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
4-(1,3-benzothiazol-2-yl)-2-({[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]amino}methyl)phenol
3-[(butan-2-yl)amino]-N-(2-ethylphenyl)propanamide