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2-{4-[1-(furan-2-ylmethyl)piperidin-4-yl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
N-[(1-benzylpiperidin-4-yl)methyl]-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
4-{4-[(5-ethylpyridin-2-yl)methyl]piperazin-1-yl}-2-methyl-6-(1H-pyrazol-1-yl)pyrimidine
N-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}-2-oxo-1,2-dihydrospiro[indole-3,3'-piperidine]-1'-carboxamide
N-[(2-fluorophenyl)methyl]-4-{4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-1-yl}benzamide
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(4-ethoxybenzoyl)piperidine
N,N-dimethyl-3-{1-[2-(methylamino)pyridine-4-carbonyl]piperidin-3-yl}propanamide
dimethyl[(4-methyl-5-{1-[4-(2-methylpropyl)benzoyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
2-amino-3-ethyl-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-cyclopropaneamido-N,4-dimethyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]benzamide
N-cyclopentyl-2-{3-[3-(pyrimidin-2-yl)phenyl]-1H-pyrazol-1-yl}propanamide
N-(1-hydroxy-3-methylbutan-2-yl)-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
(1S,5R)-6-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[3-(methylcarbamoyl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-4-oxo-1,4-dihydroquinoline-2-carboxamide
2-(2-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}-4-(pyrazin-2-yl)phenoxy)acetic acid
4-({1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]piperidin-3-yl}methyl)benzoic acid
5-butyl-1'-(4-methylpyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
ethyl 1-[(4-acetamidophenyl)methyl]-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
5-({2-benzyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
N4,N4-diethyl-6-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]pyrimidine-2,4-diamine
N4-[2-methoxy-2-(thiophen-2-yl)ethyl]-6-(morpholin-4-yl)pyrimidine-2,4-diamine
ethyl 6-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxylate
2-{3,5-dimethyl-4-[1-(3-methylbutyl)-1H-pyrazol-4-yl]-1H-pyrazol-1-yl}acetamide
3-({[1-ethyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]methyl}(methyl)amino)-1λ6-thiolane-1,1-dione
N-[1-(1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]pyridine-3-carboxamide
1-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclopropane-1-carboxamide
3-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-(methylsulfanyl)pyridine
N-[(2-chloropyridin-3-yl)methyl]-N,4-dimethyl-3-(2-oxoimidazolidin-1-yl)benzamide
2-ethyl-8-(2-phenoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]acetamide
N-(1-methyl-1H-indazol-6-yl)-3-(pyridin-3-ylmethoxy)piperidine-1-carboxamide
3-{2-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}propanoic acid
N-[3-(2-methyl-5-propylpyrimidin-4-yl)phenyl]acetamide
(3S,5S)-5-(cyclopropylcarbamoyl)-1-[4-(thiophen-2-yl)butanoyl]piperidine-3-carboxylic acid
2-(4-hydroxy-4-phenylpiperidin-1-yl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(1H-pyrrole-2-carbonyl)-1,4-diazepan-5-one
1-(cyclopropylmethyl)-N-ethyl-5-[(2-methyl-1H-indol-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-{5-[(2-aminopyridin-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-(pyrrolidin-1-yl)propan-1-one
2-{2,7-diazaspiro[4.5]decan-2-yl}pyridine-3-carboxylic acid
(3R,5S)-N-(2-methylpropyl)-5-(morpholin-4-ylmethyl)-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
3-{1-[3-(ethylcarbamoyl)phenyl]-3,5-dimethyl-1H-pyrazol-4-yl}propanoic acid
1-methyl-4-({5-[4-(1H-pyrazol-3-yl)phenyl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
2-(ethylamino)-N-[2-(2-methyl-1H-indol-1-yl)ethyl]pyrimidine-5-carboxamide
(4aS,7aR)-1-(4-chloro-2-methoxybenzoyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]acetamide
5-acetyl-N-[3-(4-methylpiperazin-1-yl)propyl]thiophene-3-carboxamide
5-[4-(2-ethoxyphenyl)piperazin-1-yl]-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
2-[2-(2,4-dimethylphenoxy)ethyl]-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
2-(dimethylamino)-2-(4-fluorophenyl)-N-[2-(pyrrolidin-1-yl)ethyl]acetamide