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2-[1-(1H-indazole-3-carbonyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazole
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-[(5-propylfuran-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
1-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-3-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}urea
methyl 4-{[4-(3,4-dichlorophenyl)piperazin-1-yl]methyl}-1H-pyrazole-3-carboxylate
1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-5-phenylpentan-1-one
1-{[3,5-dichloro-4-(propan-2-yloxy)phenyl]methyl}piperidine-4-carbonitrile
2,6,8-trimethyl-4-[3-(pyridin-3-yl)azetidine-1-carbonyl]quinoline
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)but-3-enamide
2-[(1E)-2-({4-[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)prop-1-en-1-yl]-4-chlorophenol
3-(3-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propanamide
N-methyl-2-[N-methyl-1-(1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinolin-3-yl)formamido]propanamide
1-(4-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(pyridin-4-ylmethyl)propanamide
3-methyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-1H-pyrazole-5-carboxamide
N-[5-(ethylsulfanyl)-1,3,4-thiadiazol-2-yl]-2-[4-(6-oxo-1,6-dihydropyridazin-4-yl)piperazin-1-yl]acetamide
4-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}-1-phenyl-1H-pyrazole
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}({[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
N-[(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)methyl]-4-phenylbenzamide
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-{1-[1-(2-methoxybenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
4-[5-(oxan-4-yl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
4-(3-chloro-4-fluorobenzoyl)-1-(4-methylphenyl)piperazin-2-one
(3R,4S)-4-[ethyl({[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl})amino]oxolan-3-ol
(3aR,5S,6S,7aS)-2-[(3-methyl-1,2-oxazol-5-yl)methyl]-octahydro-1H-isoindole-5,6-diol
[5-(5-ethylpyrimidin-2-yl)-7-fluoro-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-[(5-chloro-2-methoxyphenyl)methyl]-N-ethyl-3,4-dimethoxybenzamide
4-(3-cyclohexylpyrrolidine-1-carbonyl)-1-(3-phenylpropyl)-1H-1,2,3-triazole
(2R,3R,6R)-5-(2-methoxyethyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-{1-[1-(2-methoxyacetyl)piperidine-3-carbonyl]piperidin-4-yl}benzonitrile
N-[(1S,2R)-2-hydroxy-1,2-diphenylethyl]-4-methylpiperidine-4-carboxamide
(1S,5R)-6-(2-methoxyethyl)-3-(5-methyl-4-phenylthiophene-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
6-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3,5-dimethyl-1,2-oxazole-4-carboxamide
1-(cyclopropylmethyl)-5-(3-phenoxypropanoyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-[3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carbonyl]oxane-4-carbonitrile
4-[1-(2-fluorobenzoyl)piperidin-4-yl]-5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidine
4-benzoyl-6-(cyclopropylmethoxy)-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
8-fluoro-2-{[methyl(oxan-2-ylmethyl)amino]methyl}quinolin-4-ol
[(1-ethylpyrrolidin-2-yl)methyl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
1-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-4-phenylbutane-1,4-dione
2-(2-chloro-4-{[methyl(quinolin-5-ylmethyl)amino]methyl}phenoxy)acetamide
1-[(2,3-difluorophenyl)methyl]-3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)urea
(4aS,8aR)-6-(3-chlorothiophene-2-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
[(4-methyl-1H-imidazol-5-yl)methyl][(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amine
3-[(4-fluorophenyl)formamido]-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
3-methoxy-1-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1,2-dihydropyridin-2-one
[3-(3-methoxypropyl)-1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-3-yl]methanol
1-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-2-(morpholin-4-yl)ethane-1,2-dione
2,4-dimethyl-N-[(3-methylphenyl)(thiophen-2-yl)methyl]pyrimidine-5-carboxamide