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N-(2-methylpropyl)-3-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]propanamide
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-3-(1H-pyrazol-4-yl)benzamide
3-[(2-fluorophenyl)formamido]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]propanamide
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(morpholin-4-yl)benzamide
2-[2-(phenylsulfanyl)ethyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-{[4-(2-methylphenyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2-methylpropyl)-N-[3-(2-methylpyrimidin-4-yl)phenyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
2-[(2-{[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]carbamoyl}phenyl)amino]acetic acid
1-ethyl-N-({1-[(3-methylthiophen-2-yl)methyl]pyrrolidin-3-yl}methyl)-1H-pyrazole-4-carboxamide
N-methyl-5-[3-(pyridin-2-yl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
N-[2-(dimethylamino)ethyl]-N-ethyl-4-(1H-pyrazol-4-yl)butanamide
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-2-(2-chloro-4-fluorophenyl)ethan-1-one
3-(5-{2-[3-(methylsulfanyl)phenyl]acetyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
[(1-cyclopentylpiperidin-4-yl)methyl]({[4-methoxy-3-(methoxymethyl)phenyl]methyl})(oxolan-2-ylmethyl)amine
5-(4-methyl-1,4-diazepane-1-carbonyl)-2-(phenoxymethyl)pyrimidin-4-ol
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}acetamide
4-[(4-methyl-1H-pyrazol-1-yl)methyl]-N-(quinolin-5-yl)piperidine-1-carboxamide
[(3R,4R)-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
1-[2-(3-fluorophenyl)ethyl]-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-6-oxopiperidine-3-carboxamide
5-{[methyl({[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl})amino]methyl}pyrimidin-2-amine
3-{5-[(3,4-difluorophenyl)carbamoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
1-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-2-(methoxymethyl)piperidine
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(1H-pyrrole-3-carbonyl)piperidine
[4-(3,6-dimethyl-1-benzofuran-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol
naphthalen-1-yl (7S,9aR)-7-(1H-indol-3-ylmethyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
7-methyl-3-(2-phenylpropyl)-3,7,11-triazaspiro[5.6]dodecan-12-one
N-methyl-N-(2-phenylethyl)-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
5-[2-(propan-2-yloxy)phenoxy]-1-azabicyclo[3.2.1]octane
3-({1-[(2S)-1-acetylpyrrolidine-2-carbonyl]piperidin-4-yl}methyl)benzoic acid
N-ethyl-2-(4-{[4-(pyridin-3-yl)phenyl]methyl}piperazin-1-yl)acetamide
2-amino-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-6-(propan-2-yl)pyrimidine-4-carboxamide
6-(4-ethylphenyl)-N-(2-hydroxyethyl)-N-propylimidazo[2,1-b][1,3]thiazole-3-carboxamide
9-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
5-(2,6-dimethylbenzoyl)-3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
(1S,5R)-3-benzyl-6-[(2,5-dimethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
4-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-1-[(4-methoxyphenyl)methyl]piperazin-2-one
2-{4-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazin-1-yl}acetic acid
3-{[4-(methylamino)pyrimidin-2-yl]amino}-N-(2-methylphenyl)propanamide
2-(morpholin-4-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]benzamide
(3S,4R)-3-ethyl-4-methyl-1-{thieno[2,3-d]pyrimidin-4-yl}piperidin-4-ol
2-[methyl({5-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]ethan-1-ol
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-3-(1-methyl-1H-pyrrol-2-yl)propan-1-one
3-(2-amino-1,3-thiazol-4-yl)-N-{2-[3-(trifluoromethyl)phenyl]ethyl}propanamide
N-[2-(3,5-dimethoxyphenyl)ethyl]-4-methylpyrimidine-5-carboxamide
N-{2-methoxy-4-[(E)-2-phenylethenyl]phenyl}acetamide
2-amino-5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-6-(thiophen-2-yl)pyridine-3-carbonitrile
1-[(1-propyl-1H-imidazol-2-yl)methyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
4-[(2-fluorophenyl)methyl]-3-[2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-oxoethyl]piperazin-2-one
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}butan-1-one