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(1S,5R)-6-benzyl-3-(3-methanesulfonylpropanoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(3S,4R)-1-(1H-imidazol-2-ylmethyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-N-[2-(thiophen-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(3S,4R)-1-[2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
3-(2-chlorophenyl)-3-phenyl-1-[4-(pyrrolidin-1-yl)piperidin-1-yl]propan-1-one
3-(2-hydroxyphenyl)-N-[(2-methoxyphenyl)methyl]-N-propylpropanamide
2-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-oxoacetamide
N-[(5-chloro-2-propoxyphenyl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]-2-methyl-1,3-thiazole-4-carboxamide
N-methyl-3-[methyl({[4-(5-methylfuran-2-yl)phenyl]methyl})amino]butanamide
3-[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-ol
2-(3-chlorophenyl)-N,N-dimethylbenzamide
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(methylsulfanyl)propan-1-one
(1R,5S,6R)-3-{[2-(methylsulfanyl)phenyl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-methyl-1H-imidazole-4-sulfonamide
N-ethyl-2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidin-4-amine
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N,6-dimethyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
5-{[2-(dimethylamino)-2-(2-methylphenyl)acetamido]methyl}-N-methylfuran-2-carboxamide
[4-({methyl[(5-phenylthiophen-2-yl)methyl]amino}methyl)oxan-4-yl]methanol
3-benzyl-4-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[(5-methylfuran-2-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
1-[(3S,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-4-(thiophen-2-yl)butan-1-one
(2R,6R)-11-methoxy-4-(1-methylpiperidin-4-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
5-[2-(2-methoxyethyl)piperidine-1-carbonyl]-2-(3-phenylpropyl)-1,3-benzoxazole
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
4-hydroxy-2-(pyridin-2-yl)-N-{3-[(pyridin-3-yl)amino]propyl}pyrimidine-5-carboxamide
8-(1H-imidazol-2-ylmethyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1S,5R)-6-[5-(ethylsulfanyl)thiophene-2-carbonyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
3-(2-amino-1,3-thiazol-4-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]propan-1-one
N-methyl-5-({[4-(piperidin-3-yl)phenyl]formamido}methyl)-1,2,4-oxadiazole-3-carboxamide
4-phenyl-5-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrimidin-2-amine
N-(2H-1,3-benzodioxol-5-yl)-1-[(4-fluoro-2-methoxyphenyl)methyl]piperidin-3-amine
{3-[(3-chlorophenyl)methyl]-1-(pyridine-3-sulfonyl)piperidin-3-yl}methanol
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methanesulfonylethan-1-one
2-(3-fluorophenyl)-1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidine
N-(2-methoxyethyl)-2-(4-phenylpiperidin-1-yl)-N-(thiophen-3-ylmethyl)acetamide
(3aR,6aS)-1-oxo-5-[(3-phenoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-{4-[(3S,4R)-3-cyclopropyl-4-[(2-methylpyrimidin-4-yl)amino]pyrrolidin-1-yl]piperidin-1-yl}ethan-1-one
2-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane-9-carbonyl}pyridin-4-amine
3-({1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}methyl)benzoic acid
1-(4-methoxyphenyl)-4-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}butane-1,4-dione
4-(3-methyl-1,2,4-oxadiazol-5-yl)-2-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridine
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-{[3-(difluoromethoxy)phenyl]methyl}urea
1-{2-[(isoquinolin-5-ylmethyl)(methyl)amino]pyrimidin-4-yl}pyrrolidin-3-ol
8-(6-aminopyrimidin-4-yl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(2-phenyl-1H-imidazol-1-yl)-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}acetamide
1,3-dimethyl-4-[6-methyl-2-(1H-pyrazol-4-yl)quinoline-4-carbonyl]piperazin-2-one
2-(2-chloro-6-fluorophenyl)-1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine