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N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-5-propyl-1,3,4-oxadiazol-2-amine
1-cyclopentyl-N-methyl-N-[3-(2-methylphenoxy)propyl]-5-oxopyrrolidine-3-carboxamide
1-(2-hydroxyethyl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
1-[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]piperidine-4-carboxamide
1-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1-methyl-3-[2-(propan-2-yl)-1H-1,3-benzodiazol-5-yl]urea
1-[(4aR,8aR)-6-[2-(2-methoxyphenyl)acetyl]-decahydro-1,6-naphthyridin-1-yl]-2-cyclopentyl-2-phenylethan-1-one
N-{[7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
4-(cyclopropylmethyl)-N-[2-fluoro-5-(trifluoromethyl)phenyl]-3-(2-hydroxyethyl)piperazine-1-carboxamide
methyl 6-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}pyridine-2-carboxylate
1-(2-methoxyacetyl)-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]piperidine-3-carboxamide
2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-4H-chromen-4-one
N-[3-(3-fluorophenyl)phenyl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
N-methyl-2-{3-[2-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]phenyl}acetamide
N-[2-(5-methyl-1,3-oxazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-3-(4-methylphenyl)propanamide
1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-4-phenylpyrrolidin-2-one
N-[(3R,4S)-4-cyclopropyl-1-(3-hydroxypropyl)pyrrolidin-3-yl]-2-(5,5-dimethyl-2,4-dioxoimidazolidin-1-yl)acetamide
1-[2-({[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}(methyl)amino)ethyl]piperidin-2-one
N-{2-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-2-oxoethyl}methanesulfonamide
3-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]urea
N-(propan-2-yl)-1-[(1s,4s)-4-[3-(4-methoxyphenyl)propanamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-N,N-dimethylaniline
6-(2-chlorophenyl)-7-(cyclopropylmethyl)-2-[(3R)-3-hydroxypyrrolidine-1-carbonyl]-7H,8H-imidazo[1,2-a]pyrazin-8-one
dimethyl({2-[2-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]ethyl})amine
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N,4-dimethyl-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
3-(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine-1-carbonyl)pyridazine
5-acetyl-N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)thiophene-3-carboxamide
N-[1-(1H-imidazol-1-yl)butan-2-yl]-2-(3-methyl-1,2-oxazol-5-yl)acetamide
N-{[2-(4-acetylpiperazin-1-yl)-6-methylquinolin-3-yl]methyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]-2-methylpropanamide
[(1-methylpiperidin-4-yl)methyl]({[2-(methylsulfanyl)pyrimidin-5-yl]methyl})(2-phenylethyl)amine
3-[1-(2,3-dihydro-1H-inden-5-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-6-methyl-1,2-dihydropyridin-2-one
1-{2-oxo-2-[(3S,4R)-3-propyl-4-[(pyrimidin-2-yl)amino]pyrrolidin-1-yl]ethyl}imidazolidine-2,4-dione
6-methoxy-3-methyl-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1-benzofuran-2-carboxamide
N'-(3-chloro-4-fluorophenyl)-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]propanediamide
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
N-[2-(dimethylamino)ethyl]-5-(9H-purin-6-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidine
5-(5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(1s,4s)-4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]cyclohexan-1-ol
5-[(4-fluorophenyl)methyl]-5-(piperidin-4-yl)-3-(pyrazin-2-ylmethyl)imidazolidine-2,4-dione
6-[4-(hydroxymethyl)phenyl]-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
3-[(4aR,7aS)-4-[(5-chlorothiophen-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}({[3-(3-fluorophenyl)oxolan-3-yl]methyl})methylamine
4-[1-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidin-3-yl]benzoic acid
(1R,5R)-6-(cyclobutylmethyl)-3-(2-phenylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3,5-dimethyl-4,5-dihydro-1,2-oxazole-5-carboxamide
N-(4-{[2-(hydroxymethyl)azepan-1-yl]methyl}phenyl)acetamide
5-{[1-(4-chlorophenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazole
3-[(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)methyl]benzonitrile
1-{[(2S,4S)-4-fluoro-1-{2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carbonyl}pyrrolidin-2-yl]methyl}-3,3-dimethylurea
4-[(3-fluorophenyl)methyl]-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,4-diazepan-5-one