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2-({2-[4-(1H-imidazol-1-yl)phenyl]-1H-imidazol-1-yl}methyl)-4,6-dimethylpyrimidine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-cyclopentyl-2-{[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]amino}propanamide
1-({3-[3-(3-methoxypropyl)piperidine-1-carbonyl]phenyl}methyl)azepane
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)amine
4-(3-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methoxy}phenyl)morpholine
1-(1,3-benzoxazol-2-yl)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}piperidin-4-amine
2-[N-(4-methylphenyl)methanesulfonamido]-N-[(5-methylpyrazin-2-yl)methyl]acetamide
3-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-1-(2-methyl-1-benzofuran-7-yl)urea
propyl 7-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinoline-2-carboxylate
2-acetamido-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)acetamide
5-(2-fluorophenoxymethyl)-N-[(3-methyl-1-benzofuran-2-yl)methyl]-1H-pyrazole-3-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-methylpyrido[2,3-d]pyrimidin-4-amine
5-(2-carbamoylethyl)-N-cyclopentyl-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[(3-ethyl-1,2-oxazol-5-yl)methyl]-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
1-(2-chloroprop-2-en-1-yl)-6,7-dimethoxy-3-[({[3-(trifluoromethyl)phenyl]methyl}amino)methyl]-1,2-dihydroquinolin-2-one
1-{3,5-dimethyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-pyrrol-2-yl}ethan-1-one
(3R,4S)-4-[4-(2,6-dimethylquinoline-4-carbonyl)-1,4-diazepan-1-yl]oxolan-3-ol
N-[2-(1H-pyrazol-1-yl)ethyl]-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-3,5-dimethyladamantane-1-carboxamide
1-{3-[(2-methylphenyl)methoxy]azetidin-1-yl}-3-(1-methylpiperidin-3-yl)propan-1-one
2-(4-fluoro-3-methylphenyl)-2-[(furan-2-ylmethyl)(pyridin-2-ylmethyl)amino]acetic acid
2-(2-ethyl-1H-imidazol-1-yl)-1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-methyl-3-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrazine
2-({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}(methyl)amino)-N-methylacetamide
2-[(1S,5R)-3-(1-benzofuran-2-ylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-cyclopropyl-3-{1-[4-(dimethylamino)benzoyl]piperidin-3-yl}propanamide
(4aS,7aR)-4-benzyl-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-sulfonamide
1-{1-[6-(1H-indol-6-yl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
2-(3-methoxypropyl)-9-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-2,9-diazaspiro[5.5]undecan-3-one
1-[7-(3-chlorophenyl)-9-[(1-methylpiperidin-3-yl)methoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(4-fluorophenyl)ethan-1-one
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(pyridin-2-ylmethyl)piperazine
5-[4-(3-methoxyphenyl)piperazine-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
N,N-dimethyl-5-[(1-methyl-1H-indol-3-yl)methyl]-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
2-(5-{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]pyrrolidin-2-yl}-1,2,4-oxadiazol-3-yl)pyridine
3-(2-hydroxyethyl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]-1-{3-[(trifluoromethyl)sulfanyl]phenyl}urea
N-[(5-fluoro-2,3-dimethyl-1H-indol-7-yl)methyl]-2-(1H-imidazol-1-yl)acetamide
N-[(3R,4R)-3-hydroxy-1-[3-(piperidin-1-yl)propanoyl]piperidin-4-yl]pyrazine-2-carboxamide
2-(oxolan-2-ylmethyl)-4-[3-(4-phenylpiperazine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N,2-dimethyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(thiophen-2-ylformamido)propanamide
2-{4-[(3ar,6ar)-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]piperazin-1-yl}pyrazine
1-[3-({[(1-methylpiperidin-4-yl)methyl](2-phenylethyl)amino}methyl)phenyl]ethan-1-one
N-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(oxolan-2-ylmethyl)propanamide
2-[4-chloro-2-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]acetic acid
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(pyrazine-2-carbonyl)piperidine-2-carboxamide
(2S)-3-methyl-2-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}formamido)butanamide
2-butyl-8-(2-phenoxyacetyl)-2,8-diazaspiro[5.5]undecan-3-one