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1-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}piperidin-4-ol
4-(3-fluorophenoxy)-1-(1,3-thiazol-2-yl)piperidine-4-carboxylic acid
N-[(3-fluorophenyl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N,4-dimethyl-N-[2-(pyrrolidin-1-ylmethyl)propyl]quinazolin-2-amine
8-(3-methoxypyrazin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-chloro-2-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-5-(trifluoromethyl)pyridine
3-{[2-(1H-imidazol-1-yl)ethyl]sulfamoyl}-N-(oxolan-2-ylmethyl)benzamide
4-cyclopentyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}pyrimidin-2-amine
2-[2-(3,6-dimethyl-1-benzofuran-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]acetic acid
9-(4-methylpyrimidine-5-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(1,3-benzothiazol-2-yl)propyl]piperidin-3-amine
1-[(2,4-dimethoxyphenyl)methyl]-3-propoxypiperidine
(4S)-1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,3,4-trimethylpiperidin-4-ol
(4aR,7aS)-1-(2-methylpropanoyl)-4-(naphthalene-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
4-{1-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]azetidin-3-yl}pyridine
4-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]benzamide
8-methoxy-2-({2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)quinoline
3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-8-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-amino-6-(furan-2-yl)-4-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
methyl 4-{[(3S)-3-(tert-butylcarbamoyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]methyl}-1H-pyrazole-3-carboxylate
2,5-dimethyl-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
5-(2-methoxyacetamido)-1-methyl-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)-1H-imidazole-5-carboxamide
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-2-fluoro-4-methylbenzamide
1-(5-ethyl-1H-pyrrole-2-carbonyl)-4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
7-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
(3R,4R)-1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-3-cyclobutyl-4-methylpyrrolidin-3-ol
7-(cyclobutylmethyl)-2-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-2,7-diazaspiro[4.5]decan-6-one
(2S,4S,5R)-4-[(1-carboxy-1-methylethyl)carbamoyl]-5-(3-chlorophenyl)-1-methylpyrrolidine-2-carboxylic acid
N-[4-(3-methoxyphenyl)phenyl]-1-(oxane-4-carbonyl)piperidine-3-carboxamide
3-ethynyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
2-{1-[2-(2,5-dimethoxyphenyl)acetyl]pyrrolidin-3-yl}benzoic acid
1-(1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-4-yl)-3-(pyrrolidine-1-carbonyl)piperidine
4-(hydroxymethyl)-1-[4-(4-hydroxyphenyl)benzoyl]azepan-4-ol
N-(2-methoxyethyl)-2-methyl-N-propylthieno[2,3-d]pyrimidin-4-amine
N-{[4-(but-2-yn-1-yloxy)phenyl]methyl}-N-cyclopentylthiophene-2-carboxamide
(2R,3R,6R)-5-(1H-imidazole-2-carbonyl)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(3-methylphenyl)-3-{[1-(2-methylpropyl)piperidin-4-yl]amino}propanamide
(3S,4S)-3-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-4-hydroxy-1λ6-thiolane-1,1-dione
1-[4-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)-1,4-diazepan-1-yl]ethan-1-one
methyl 8-cycloheptyl-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
N-(3-acetamido-4-fluorophenyl)-4-(4H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methylbenzamide
5-cyclobutanecarbonyl-1'-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
8-(cyclopentylmethyl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
5-{[benzyl(methyl)amino]methyl}-N-[1-(6-methylpyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
2-methoxy-1-(1'-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one