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1-cycloheptyl-N-[2-(5-methylfuran-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
[5-({[2-(dimethylamino)ethyl][(3-methylthiophen-2-yl)methyl]amino}methyl)furan-2-yl]methanol
3-(2-methoxyethyl)-1-(morpholine-4-carbonyl)piperidine-3-carboxylic acid
N-[1-(3-phenylpropyl)piperidin-3-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-(5-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)phenol
3-{[(cyclopropylmethyl)(propan-2-yl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-[4-({[(1R,2S)-2-hydroxycyclohexyl](methyl)amino}methyl)phenoxy]-1-(morpholin-4-yl)ethan-1-one
(2-methoxyethyl)(methyl){[1-phenyl-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}amine
2-[2-(4-fluorophenyl)acetyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-{[1-(7-methoxy-4-methylquinolin-2-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
5-[(2S)-1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)pyrrolidin-2-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
2,3,5,6-tetramethyl-N-[2-(2-oxoimidazolidin-1-yl)ethyl]benzamide
6-[3-(3-fluorophenoxymethyl)piperidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(1-methyl-1H-pyrrol-3-yl)-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]({2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl})amine
N-[3-methyl-1-(pyridin-3-yl)butyl]-1,4-dithiepan-6-amine
2-(morpholin-3-yl)-N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}acetamide
5-[2-(2-aminoethyl)morpholin-4-yl]-2-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-2,3-dihydropyridazin-3-one
(3S)-N-tert-butyl-2-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(2R)-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-hydroxy-N-methyl-2-phenylacetamide
1-(2-methoxyphenyl)-3-(1-{1-[2-(methylamino)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
7-methyl-2-{3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanoyl}-2,7-diazaspiro[4.5]decan-6-one
ethyl(2-methoxyethyl){[1-methyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]methyl}amine
3-ethyl-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}urea
(4aS,7aR)-1-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-(methoxymethyl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]pyrimidin-4-amine
2-[4-(4-chloro-1H-indazol-1-yl)phenyl]-N-methylacetamide
3-(2-acetylphenyl)-4-methyl-1,2-dihydroquinolin-2-one
2-[4-(1-cyano-1-methylethyl)phenyl]-2-[methyl(oxan-4-ylmethyl)amino]acetic acid
[(1-ethyl-1H-pyrazol-4-yl)methyl](methyl){[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}amine
1-[(2-fluorophenyl)methyl]-4-{1H-pyrrolo[2,3-b]pyridin-6-yl}-1,4-diazepane
2-amino-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-fluoro-N,3-dimethyl-1-benzofuran-2-carboxamide
(1R,5S)-6-methyl-3-(5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2-acetyl-1H-1,3-benzodiazol-1-yl)-N-(1-benzyl-1H-pyrazol-3-yl)acetamide
{3-[2-(1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]propyl}dimethylamine
1-benzyl-5-(4-benzylpiperidine-1-carbonyl)-N-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carboxamide
2-{[(2,2-dimethyloxan-4-yl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]propanamide
2-methyl-5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-3,4-dihydropyrimidin-4-one
ethyl 2-{1-[4-(propan-2-yl)benzoyl]piperidin-2-yl}acetate
6-fluoro-2-{[2-(1,3-thiazol-2-yl)piperidin-1-yl]methyl}quinoline
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(1H-pyrazol-1-yl)benzamide
(1S,5R)-3-[(4-fluoro-3-methoxyphenyl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 2-[methyl({[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl})amino]acetate
N-methyl-2-(methylamino)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,3-thiazole-4-carboxamide
3-{[1-(ethylsulfanyl)propan-2-yl]amino}-1-(4-methylpiperidin-1-yl)propan-1-one
2-(azetidine-1-carbonyl)-5-chloro-3-phenyl-1H-indole
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-methyloxane-2-carboxamide
2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decane