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2-(4-{[2-(2-methylpropyl)morpholin-4-yl]methyl}phenoxy)acetic acid
1-[1-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)piperidine-2-carboxamide
2-[2-({2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}methyl)phenoxy]propanoic acid
5-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,2-dihydropyridin-2-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-methoxypyridine-4-carboxamide
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
2-methyl-6-[2-(pyridin-3-yl)piperidine-1-carbonyl]-2,3-dihydropyridazin-3-one
3-benzyl-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}pyrrolidine
N-{[(3S,4S)-3-hydroxy-1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidin-4-yl]methyl}benzamide
N-(2-methoxyethyl)-3-[(naphthalen-1-ylformamido)methyl]piperidine-1-carboxamide
2-[5-(1H-indol-2-yl)-4-phenyl-1H-imidazol-1-yl]-1-(pyridin-3-yl)ethan-1-ol
[(4-chloro-1-methyl-1H-indazol-3-yl)methyl](methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
2-ethyl-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]pyrimidine-5-carboxamide
[({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)sulfamoyl]dimethylamine
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-(2,3-dimethyl-1H-indole-7-carbonyl)-2-azaspiro[4.4]nonane
1-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
1-[5-({[2-(dimethylamino)ethyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
3-[3-(1H-imidazol-1-yl)propyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{2-oxo-4-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]piperazin-1-yl}benzonitrile
3-(2-chlorophenyl)-N-cyclopropyl-3-(3-hydroxyphenyl)propanamide
3-[(4aS,8aR)-decahydroisoquinolin-2-ylmethyl]-N-(1-methyl-1H-1,2,4-triazol-3-yl)benzamide
{4-[(2,3-dichlorophenyl)methyl]-1-methylpiperazin-2-yl}methanol
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-2-(2-methyl-1,3-thiazol-4-yl)acetamide
(3ar,6ar)-N-[3-(pyridin-2-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
ethyl 3-benzyl-1-[(propan-2-yl)carbamoyl]piperidine-3-carboxylate
[1-({methyl[4-(propan-2-yl)pyrimidin-2-yl]amino}methyl)cyclobutyl]methanol
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)furan-2-carboxamide
2-(2-phenylethyl)-9-(pyrimidin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-(5-{[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
1-cyclopropyl-5-oxo-N-[1-(pyrazin-2-yl)piperidin-4-yl]pyrrolidine-3-carboxamide
(3S,4S)-4-cyclopropyl-1-{[2-(ethylamino)pyrimidin-5-yl]methyl}pyrrolidine-3-carboxylic acid
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)propanamide
7-cyclohexyl-2-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrimidin-2-amine
2-(dimethyl-1,3-thiazol-5-yl)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}acetamide
1-{2-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}azepan-2-one
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-methoxyphenyl)-3-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}urea
N,1,3-trimethyl-2,6-dioxo-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(3-hydroxypiperidin-1-yl)ethan-1-one
ethyl 4-[(4-methoxyphenyl)methyl]-1-[2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetyl]piperidine-4-carboxylate
1-(2,2-dimethylpropyl)-3-hydroxy-3-({[(5-methylpyrazin-2-yl)methyl]amino}methyl)piperidin-2-one
8-[2-(4-fluoro-3-methylphenyl)acetyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(2-ethyl-1,3-thiazol-4-yl)methyl]-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
2-[2-methyl-3-({[3-(3-oxopiperazin-1-yl)propyl]amino}methyl)-1H-indol-1-yl]acetamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1H-imidazol-2-ylmethyl)acetamide
{3-[(4-fluorophenyl)methyl]-1-[1-(2-methylphenyl)piperidin-4-yl]piperidin-3-yl}methanol
2-amino-4-{2-[2-(dimethylamino)ethoxy]phenyl}-6-(propan-2-yl)pyridine-3-carbonitrile