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2-ethyl-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
(2R,3R,6R)-5-cyclobutanecarbonyl-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(piperidin-1-yl)-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)acetamide
(2S,4R)-4-hydroxy-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)pyrrolidine-2-carboxamide
N-{2-[(4-chlorophenyl)methoxy]ethyl}-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
1-[(3-methoxyphenyl)methyl]-4-(6-methoxypyrimidin-4-yl)piperazin-2-one
4-(5-methylfuran-2-yl)-N-[(1R,3S)-3-(pyrrolidine-1-carbonyl)cyclopentyl]benzamide
6-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]-1H-indole
2-(1-methyl-1H-imidazol-2-yl)-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine
N-[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
N-methyl-N-(quinolin-8-ylmethyl)-9H-purin-6-amine
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-2-(morpholin-2-yl)acetamide
4-{5-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]-1H-pyrazol-3-yl}phenol
7-[2-hydroxy-4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
[3-(2-methoxyethyl)-1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl]methanol
3-hydroxy-3-({[2-(1H-imidazol-4-yl)ethyl]amino}methyl)-1-(2-phenylethyl)piperidin-2-one
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-(4-methylphenoxy)piperidine-4-carboxamide
3-chloro-5-[4-(2,3-dihydro-1H-inden-2-yl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
(1S,5R)-3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4,6-dimethyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-({7-[2-(2,5-dimethoxyphenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)pyrazine-2-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-1-{spiro[azepane-4,2'-chromene]-1-yl}propan-1-one
2-{ethyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino}ethan-1-ol
2-(1-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)-5-fluoro-1H-1,3-benzodiazole
4-{[1-(3-fluorophenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}piperazin-2-one
2-[4-(6-aminopyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]pyridine-3-carbonitrile
(3S,4S)-N-[2-(4-fluorophenoxy)pyridin-3-yl]-3-hydroxy-4-(propan-2-yloxy)pyrrolidine-1-carboxamide
3-[2-(azetidin-1-yl)-2-oxoethyl]-1-[(4-fluorophenyl)methyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-methyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-methyl-3-(2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-1-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}urea
2-(ethoxymethyl)-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]ethan-1-one
1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-N-(2-methylprop-2-en-1-yl)piperidine-4-carboxamide
2-(1-ethylpiperidin-4-yl)-N-methyl-N-(1H-pyrazol-3-ylmethyl)acetamide
(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethyl-N-[4-(methylsulfanyl)phenyl]piperidine-1-carboxamide
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N,N-dimethyl-2-[(1S,5R)-6-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
2-[4-(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)-6-methylpyrimidin-2-yl]phenol
(1S,5R)-6-(cyclobutylmethyl)-3-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
5-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
N-methyl-N-[2-(pyridin-2-yl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-(naphthalen-1-ylmethyl)piperazin-2-one
(2R,6R)-4-{[4-(methylcarbamoyl)phenyl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
[(1-cyclopentylpiperidin-4-yl)methyl]({[2-(methylsulfanyl)pyrimidin-5-yl]methyl})(oxolan-2-ylmethyl)amine
2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-4-carbonitrile
1-(4-phenyl-1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperidin-4-yl)ethan-1-one
1-[(3,5-dimethylphenyl)methyl]-4-(3-ethyl-1H-pyrazole-4-carbonyl)piperazin-2-one