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6-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)-2-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)-1,2,3,4-tetrahydro-2,7-naphthyridine
N-[(2,6-difluorophenyl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(4aR,7aS)-1-(2-methylpropyl)-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
propyl 4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[1-(pyridin-4-yl)propyl]butanamide
2-[5-({5-[morpholin-4-yl(phenyl)methyl]-1H-1,2,3,4-tetrazol-1-yl}methyl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
2-[(3,5-difluorophenyl)methyl]-8-[(2S)-2-(methylamino)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
(1R,2R)-2-phenyl-N-{2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}cyclopropane-1-carboxamide
4-{[4-(3-methoxyphenyl)-2-methyl-3-oxopiperazin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
(1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methanol
2-[(4-chlorophenyl)methyl]-8-(1H-pyrrole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
[(1R,3S,3aS,6aR)-5-ethyl-3-(5-fluoro-2-methoxyphenyl)-1-(2-methylpropyl)-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methylpiperazine-1-carboxamide
1-[1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-oxo-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1-oxaspiro[4.5]decane-4-carboxamide
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-({[5-(methoxymethyl)furan-2-yl]formamido}methyl)benzoate
2-{9-[2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
(1,4-dioxan-2-ylmethyl)(7-methoxy-3,7-dimethyloctyl)amine
methyl 1-(2-methoxyethoxy)-2-oxo-8-[2-(1H-pyrazol-1-yl)benzoyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(methylamino)pyridine-4-carboxamide
N3-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[3-(morpholin-4-yl)propyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
N-[2-(dimethylsulfamoyl)ethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1-(3-methanesulfonamidophenyl)urea
4-methyl-6-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrimidin-2-amine
4-[(1-methoxypropan-2-yl)amino]-N,5-dimethyl-N-(1,2-oxazol-3-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
(2S)-4-methanesulfonyl-2-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]formamido}butanoic acid
1-[7-(6,7-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-phenylethan-1-one
(2H-1,3-benzodioxol-5-ylmethyl)(oxolan-3-ylmethyl)(pyridin-3-ylmethyl)amine
1-(piperidin-4-yl)-4-(quinolin-5-ylmethyl)-1,4-diazepan-6-ol
[(1-cyclopentylpiperidin-4-yl)methyl]({[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl})(pyridin-3-ylmethyl)amine
3-(4-fluorophenyl)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-3-phenylpropanamide
methyl 2-[8-(3-hydroxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carboxylate
1-[benzyl(methyl)amino]-3-(4-{[methyl(oxan-4-yl)amino]methyl}phenoxy)propan-2-ol
2-(5-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridin-3-yl}-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl)ethan-1-ol
4-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-6-methoxypyrimidin-2-amine
N,N-dimethyl-3-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}pyrazin-2-amine
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(1-methyl-2-oxopyrrolidin-3-yl)benzamide
(1S,5R)-N-(2,5-dimethylphenyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
(1S,5R)-6-[(dimethylcarbamoyl)methyl]-N-(3,5-dimethylphenyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1'-(1H-indazole-3-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-(2-methoxyphenoxy)ethan-1-one
1-cyclohexyl-N3-methyl-4-oxo-N5-[2-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(2-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-1,3-thiazol-4-yl)methanol
N,2-dimethyl-N-{2-[4-(propan-2-yl)phenoxy]ethyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
(2S,4S)-4-amino-1-(4-amino-6-fluoroquinoline-3-carbonyl)-N-methylpyrrolidine-2-carboxamide
N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-4-(1H-pyrazol-1-yl)benzamide
N-(3-chlorophenyl)-2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-(2-methoxy-5-methylphenyl)-2-(1,4-oxazepan-4-yl)acetic acid