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(3ar,6ar)-N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-benzyl-4-(2,5-dimethoxyphenyl)-4H-1,2,4-triazole
2-{methyl[(4-methyl-5-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amino}ethan-1-ol
1-[2-(dimethylamino)-6-[(1-methyl-1H-pyrazol-4-yl)methyl]-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
1,9-dimethyl-4-{[5-methyl-1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1,4,9-triazaspiro[5.5]undecane
4-({[4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}methyl)benzene-1-sulfonamide
1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-2-[4-(propan-2-yl)morpholin-2-yl]ethan-1-one
N-ethyl-5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-N-methylpyridin-2-amine
[(3S,5R)-5-(morpholin-4-ylmethyl)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl]methanol
5-[3-(dimethyl-1,2-oxazol-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-N,4-dimethyl-1,3-thiazol-2-amine
N-(4-{[3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazin-1-yl]methyl}phenyl)acetamide
[1-({1-[(4-methoxy-2-methylphenyl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
2-(1-methyl-1H-pyrrol-2-yl)-2-oxo-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]acetamide
N3-[2-(4-propoxyphenyl)ethyl]piperidine-1,3-dicarboxamide
ethyl 3-[(3-methoxyphenyl)methyl]-1-(prop-2-ene-1-sulfonyl)piperidine-3-carboxylate
3-{5-[1-(pyridine-2-carbonyl)piperidin-4-yl]-1,2,4-oxadiazol-3-yl}pyridazine
1-(4-butylphenyl)-3-(1H-imidazol-2-ylmethyl)urea
1-methyl-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-1H-pyrazole-4-sulfonamide
N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
1-ethyl-6-{[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]methyl}-1H-indole
(4aR,8aR)-1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-6-(3-methoxybenzoyl)-decahydro-1,6-naphthyridine
7-(2-methoxyethyl)-2-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-methoxy-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
5-(methoxymethyl)-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)thiophene-2-carboxamide
2-[(dimethylamino)methyl]-4-[1-(2-methyl-1H-1,3-benzodiazol-6-yl)-1H-imidazol-2-yl]phenol
2-cyclopropyl-5-[3-(2-fluorophenoxymethyl)piperidine-1-carbonyl]pyrimidin-4-ol
3-methyl-6-{5-[2-(1-methylpiperidin-4-yl)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
2-[4-(propan-2-yl)morpholin-2-yl]-N-[2-(pyridin-2-ylsulfanyl)ethyl]acetamide
2-({cyclopropyl[(3-ethoxyphenyl)methyl]amino}methyl)benzoic acid
N-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carboxamide
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-2-(propan-2-yloxy)propanamide
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-5-methyl-1H-indole-2-carboxylic acid
5,5-dimethyl-1-{[1-(2-methylpyridin-4-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
N-(3,5-dimethylphenyl)-3-oxo-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-({3-[4-methyl-5-(prop-2-en-1-ylsulfanyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
2-hydroxy-N-[(3R,4S)-4-(propan-2-yl)-1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}pyrrolidin-3-yl]acetamide
5-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
1-{4-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
N-[2-(4-methoxyphenyl)phenyl]-1-[(2E)-2-methylbut-2-en-1-yl]piperidine-3-carboxamide
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-1-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-3-(1-methylpiperidin-2-yl)propanamide
7-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]amino}methyl)-5-[(3-fluorophenyl)methyl]-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
1-{5H,6H-benzo[h]quinazolin-2-yl}-N,5-dimethyl-N-(oxolan-3-yl)-1H-pyrazole-4-carboxamide
3-(furan-2-yl)-4-[2-(morpholin-4-yl)pyridin-3-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
{[1-butyl-2-(cyclohexanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
(1S,6R)-3-methyl-9-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
3-{[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]methyl}-1-(1H-imidazol-2-ylmethyl)piperidine
1-[4-(2-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-2-oxoethyl)phenyl]imidazolidin-2-one
N,N-dimethyl-2-{[3-(1H-1,2,4-triazol-1-yl)adamantan-1-yl]formamido}propanamide