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methyl 4-({[5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]amino}methyl)benzoate
N-ethyl-2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-N-methylacetamide
N4-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-N2,N2,5,6-tetramethylpyrimidine-2,4-diamine
N-[3-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]carbamoyl}amino)-4-fluorophenyl]propanamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-3-ol
1-(carbamoylmethyl)-N-[(3-chloro-2-methylphenyl)methyl]piperidine-3-carboxamide
(4aR,7aS)-1-(2-hydroxyethyl)-4-(naphthalene-1-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-[3-(4-phenylbenzoyl)piperidine-1-carbonyl]quinoxaline
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1H-1,2,4-triazol-1-yl)propanamide
N-[2-methoxy-5-({[(1R,2S)-2-(methoxymethyl)cyclopentyl]carbamoyl}amino)phenyl]acetamide
N-benzyl-2-(dimethyl-1,3-thiazol-4-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
2-({2-[1-(5-ethylthiophene-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[(4-methoxyphenyl)methyl]-N-[(3-methylphenyl)methyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
(2S,4S)-4-amino-1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-N-methylpyrrolidine-2-carboxamide
N-{2-[4-(oxan-4-yl)morpholin-2-yl]ethyl}cycloheptanecarboxamide
N-ethyl-5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyrimidin-2-amine
N-{2-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-2-oxoethyl}benzamide
3-[2-(2-ethyl-1,3-benzoxazol-5-yl)ethyl]-1λ6-thiolane-1,1-dione
11-{[(2,4-difluorophenyl)methyl]amino}-4-(pyridin-4-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[(3-methylthiophen-2-yl)methyl]pyrrolidin-3-yl]-3-hydroxypropanamide
N-[1-(4-tert-butylphenyl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-{[6-chloro-4-(cyclopentylamino)quinazolin-2-yl]methyl}-3-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]propanamide
1-(4-{[3-(dimethyl-1,2-oxazol-4-yl)propyl]amino}-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)ethan-1-one
4-[4-(thiophen-2-ylmethyl)piperazin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-amine
N-methyl-1,1-dioxo-N-[(4-phenoxyphenyl)methyl]-1λ6-thiane-4-carboxamide
{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[2-(1H-imidazol-1-yl)ethyl]methylamine
N-(2-methoxyethyl)-1-{1-[(4-methylphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
2-[5-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)furan-2-yl]benzonitrile
{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(pyridin-2-yl)ethyl]amine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-8-fluoro-N-methylquinoline-2-carboxamide
2-{1-cyclohexyl-4-[(5-ethylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
3-(1-methyl-1H-imidazol-2-yl)-1-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]piperidine
1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]-2-(2H-indazol-2-yl)ethan-1-one
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-2,4-dimethyl-1,3-thiazole-5-carboxamide
2-(2-methylpropyl)-8-[4-(trifluoromethyl)pyrimidin-2-yl]-2,8-diazaspiro[4.5]decan-3-one
3-(5-fluoro-2-methoxybenzoyl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
2-[2-(dimethylamino)ethyl]-9-[2-(4-methyl-1H-pyrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-N-(pyridin-4-yl)benzamide
2,6-dimethyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]quinoline-4-carboxamide
2-oxo-N-[3-(1,3-thiazol-4-yl)phenyl]-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
2-[4-(4-methoxypyrimidin-2-yl)-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
ethyl 4-[(2S,4R)-4-aminopyrrolidine-2-amido]piperidine-1-carboxylate
4-(2-fluorophenoxy)-1-[2-(pyridin-4-yl)acetyl]piperidine-4-carboxylic acid
1-[(3-ethenylphenyl)methyl]-4-(2-methylquinolin-6-yl)piperidin-4-ol
(1-methyl-4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-2-yl)methanol
(2R,6R)-4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)propyl]-2,3,4,9-tetrahydro-1H-carbazole-6-carboxamide
2-({[1-(2-cyclohexylethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}amino)-N,N-dimethylethane-1-sulfonamide