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(2S,4R)-4-[(1-ethylpiperidin-4-yl)amino]-1-(naphthalen-1-ylmethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[1-(dimethylamino)-2-methylpropan-2-yl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(7-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1-phenylmethanesulfonamide
N-{[2-(azepan-1-yl)-7-fluoroquinolin-3-yl]methyl}-N-(2-methoxyethyl)-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{3-[3-(2-methoxybenzoyl)piperidin-1-yl]-3-oxopropyl}azepan-2-one
(3aS,6aS)-5-({2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl}methyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
{[1-butyl-2-(cyclohexanesulfonyl)-1H-imidazol-5-yl]methyl}(ethyl)(pyridin-4-ylmethyl)amine
2-(1-methyl-4-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}piperazin-2-yl)ethan-1-ol
N-(3-chloro-4-propanamidophenyl)pyridazine-3-carboxamide
4-{1-[(4-methoxyphenyl)methyl]-1H-imidazol-2-yl}-2-(propan-2-yl)-1,3-oxazole
2-(2-chlorophenoxymethyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(9H-purin-6-yl)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}piperidin-4-amine
4-(1H-1,3-benzodiazol-1-yl)-1-(9H-purin-6-yl)piperidine-4-carboxylic acid
1-methyl-N-[(1-phenylcyclopentyl)methyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-methyl-1-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}urea
(2R,3S,6R)-5-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-3-(4H-1,2,4-triazol-4-yl)benzamide
N-cyclohexyl-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-(pyridin-4-ylmethyl)acetamide
1-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2,8-dimethylquinoline-4-carboxamide
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-pyrrole-2-carboxamide
1-[1-(1-benzothiophen-2-ylmethyl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
5-({2-[5-(hydroxymethyl)furan-2-yl]-1H-imidazol-1-yl}methyl)-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-propyl-1,3-thiazole-4-carboxamide
3-benzyl-1-(3-methoxypropyl)-8-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-N-(3-methylphenyl)propanamide
N-methyl-2-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidin-4-amine
2-{[2-(3-fluorophenyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}-6-methoxyphenol
ethyl 3-[(2-fluorophenyl)methyl]-1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidine-3-carboxylate
3-{[cyclopropyl(pyridin-2-ylmethyl)amino]methyl}-N-(1-methyl-1H-1,2,3-triazol-4-yl)benzamide
3-[4-(2,3-dimethylphenyl)piperazin-1-yl]-N-(furan-2-ylmethyl)propanamide
4-(1-{1-[(5-methyl-1,2-oxazol-3-yl)methyl]piperidin-4-yl}ethyl)morpholine
2-amino-4-(2-methoxypyrimidin-5-yl)-5H-chromeno[4,3-b]pyridine-3-carbonitrile
5-(2,4-difluorophenoxymethyl)-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1,2-oxazole-3-carboxamide
5-ethyl-5-[1-(2-methoxypyrimidine-5-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
1-ethyl-7-methyl-N-{1-oxaspiro[4.4]nonan-3-yl}-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxamide
N-({3-[2-(dimethylamino)ethoxy]phenyl}methyl)-4-methyl-N-(pyridin-2-ylmethyl)benzamide
6-methyl-4-oxo-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-4H-pyran-2-carboxamide
(1R,5S,8S)-3-({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)-3-azabicyclo[3.2.1]octan-8-ol
N-{4-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-oxobutyl}acetamide
2-(4-fluoro-2-methoxyphenyl)-6-methylpyridine-3-carbonitrile
2-{2-[1-(oxolan-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]-1H-pyrrol-1-yl}pyrimidine
2-{4-[5-(4-methoxyphenyl)-1,2,4-triazin-3-yl]piperazin-1-yl}-N-(propan-2-yl)acetamide
9-methoxy-4-[5-(methoxymethyl)furan-2-carbonyl]-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1S,5R)-6-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-{[(1R,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
(1S,5R)-6-(cyclopropylmethyl)-3-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
5-(3-acetylphenoxymethyl)-N-(furan-2-ylmethyl)-N-methyl-1H-pyrazole-3-carboxamide
5-[4-(carbamoylmethyl)piperazin-1-yl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
5-chloro-4-(1-{[(2R)-1-ethylpyrrolidin-2-yl]methyl}-1H-imidazol-2-yl)-2-methoxyphenol