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(3S,4S)-1-({4-[methyl(phenyl)amino]phenyl}methyl)-4-(morpholin-4-yl)pyrrolidin-3-ol
1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
5-(2-chloro-4-methoxyphenoxymethyl)-N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
3-(2-methoxyethyl)-1-(oxan-4-yl)piperidine-3-carboxylic acid
methyl 2-chloro-4-({[1-(methylcarbamoyl)butyl]carbamoyl}amino)benzoate
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-[2-(1-methyl-1H-pyrazol-3-yl)piperidin-1-yl]ethan-1-one
(4-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}morpholin-3-yl)methanol
N-[2-(4-methoxyphenyl)ethyl]-6-methyl-N-[(1-methylpiperidin-4-yl)methyl]-4-oxo-4H-pyran-2-carboxamide
6-{2-amino-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
2-[4-(hydroxymethyl)phenyl]-N-(propan-2-yl)benzamide
3-{1-[(5-propylfuran-2-yl)methyl]azetidin-3-yl}pyridine
5-{[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2,1,3-benzoxadiazole
N-ethyl-1-(2-methoxyphenyl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazole-4-carboxamide
2-amino-4-(1-methyl-1H-pyrazol-4-yl)-6-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]pyridine-3-carbonitrile
3-[1-(4-methanesulfonylphenyl)-1H-1,3-benzodiazol-2-yl]propan-1-ol
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-(5-methyl-1,3-benzoxazol-2-yl)-decahydro-2,7-naphthyridine-2-sulfonamide
1-acetyl-N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]piperidine-4-carboxamide
5-{1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1H-imidazol-2-yl}-2-(furan-2-yl)pyrimidine
2-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-N-[(2-methoxyphenyl)methyl]acetamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
(2S,4S)-4-(benzylamino)-1-{[4-(diethylamino)phenyl]methyl}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
(2S)-1-(6-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-(methylamino)propan-1-one
N-(oxolan-2-ylmethyl)-5-(propan-2-yl)-N-(thiophen-3-ylmethyl)-1,2-oxazole-3-carboxamide
2-{4-[(2,5-dimethylphenyl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
4-(furan-2-carbonyl)-9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1S,5R)-3-[6-(3-fluorophenyl)pyridine-3-carbonyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S)-N-(2-ethyl-1H-1,3-benzodiazol-6-yl)-2-(hydroxymethyl)pyrrolidine-1-carboxamide
(3S,4S)-1-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
3-(2,5-difluorobenzoyl)-1-[3-(1H-imidazol-2-yl)benzoyl]piperidine
7-(2,2-dimethylpropyl)-2-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-2,7-diazaspiro[4.5]decane
N-ethyl-5-{[(1R,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyrimidin-2-amine
N-methyl-5-(morpholin-4-ylmethyl)-N-(3-phenylpropyl)-1,2-oxazole-3-carboxamide
5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-[(3-hydroxypyrrolidin-3-yl)methyl]-1,2-oxazole-3-carboxamide
1-{1-[2-(difluoromethoxy)benzoyl]piperidin-4-yl}-3-methylbutan-1-ol
3-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-N,N-dimethylpropanamide
[(3-ethyl-1,2-oxazol-5-yl)methyl](1H-imidazol-2-ylmethyl)methylamine
(3S,4R)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-3-methoxypiperidin-4-amine
(4aS,7aS)-6-(5-chloronaphthalene-1-carbonyl)-octahydro-1H-pyrrolo[3,4-b]pyridine
6-methyl-5-[5-(quinolin-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-2-(4-phenylphenyl)acetamide
2-(6-ethyl-4-methylquinolin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-(cyclohexylmethyl)-3-hydroxy-3-{[4-(methoxymethyl)piperidin-1-yl]methyl}piperidin-2-one
2-(5,5-dimethyl-2,4-dioxoimidazolidin-1-yl)-N-[2-(7-methyl-1H-indol-3-yl)ethyl]acetamide
2-methoxy-3-{[(propan-2-yl)amino]methyl}-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-(azetidine-1-carbonyl)-N-[2-(pyridin-2-yl)ethyl]benzene-1-sulfonamide
2-{4-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]piperidin-1-yl}acetamide
8-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
(1-{[6-(4-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-2,5-dihydro-1H-pyrrol-2-yl)methanol
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-{4-[(5-methylfuran-2-yl)methyl]morpholin-3-yl}acetamide