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2-(furan-2-yl)-1-(pyrrolidine-1-carbonyl)azepane
1-({3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
7-(7-chloro-4-hydroxyquinoline-3-carbonyl)-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(2,1,3-benzothiadiazol-5-ylmethyl)-N-(3-fluorophenyl)piperidin-3-amine
4-{[(3S,5R)-1-(2-phenylethyl)-5-(pyrrolidine-1-carbonyl)piperidin-3-yl]methyl}morpholine
4-(pyridin-3-yl)-N-{[1-(pyrrolidin-1-yl)cyclopentyl]methyl}pyrimidin-2-amine
1-{[2-(difluoromethoxy)phenyl]methyl}-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N3-cycloheptyl-N5-[1-(furan-2-yl)ethyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-hydroxy-2-(pyridin-4-yl)-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrimidine-5-carboxamide
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)acetamide
N-[3-(1H-imidazol-1-yl)propyl]-3-[(2-phenylethyl)amino]-5-(pyrrolidine-1-sulfonyl)benzamide
N-[4-(dimethylamino)phenyl]-3-[(1-hydroxypropan-2-yl)amino]propanamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
2-{4-[(3-chlorophenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
N-[(4-ethoxyphenyl)methyl]-2-methanesulfonyl-N-(2-methoxyethyl)acetamide
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-[(3-methylthiophen-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
5-(oxolan-2-yl)-N-[1-(thian-4-yl)piperidin-4-yl]thiophene-2-carboxamide
6-[(2S)-2,4-dimethyl-3-oxopiperazin-1-yl]-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-3-(4H-1,2,4-triazol-4-yl)benzamide
N-benzyl-6-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-6-azaspiro[2.5]octane-1-carboxamide
({5-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylthian-4-amine
9-{[4-(3-hydroxyprop-1-yn-1-yl)phenyl]methyl}-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-(3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl)ethan-1-one
1'-(5-propyl-1,2-oxazole-3-carbonyl)-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
(4aR,7aS)-1-benzyl-4-(1,3-thiazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-N,N-dimethylpiperazine-1-sulfonamide
1-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-[(2R)-3-methylbutan-2-yl]urea
7-fluoro-2-(2-methylpyrimidin-5-yl)-4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)quinoline
2-(propan-2-yl)-4-({4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)pyrimidine
1-{1-[(2-aminopyridin-3-yl)methyl]piperidin-4-yl}-2-phenylethan-1-ol
4-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-3-(3-fluorophenyl)piperazin-2-one
{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
2-(3-phenylpropyl)-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,8-diazaspiro[4.5]decan-3-one
N-{1-[4-(dimethylamino)phenyl]propan-2-yl}-4-methylpyrimidin-2-amine
2-[(cyclopropylmethyl)(propyl)amino]-2-[4-(propan-2-yloxy)phenyl]acetic acid
(2E)-1-(3-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-3-(2,5-difluorophenyl)prop-2-en-1-one
2-(2-methyl-1-{4-[1-(propan-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-1-yl}propyl)pyridine
N-[(3-methoxyphenyl)methyl]-3-[1-(pyridazine-4-carbonyl)piperidin-3-yl]propanamide
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(4-fluorophenyl)piperazine
5-benzyl-4-ethyl-1-(4-methylphenyl)piperazin-2-one
9-(2,8-dimethylquinoline-3-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
1-[3-(4-chlorophenyl)propyl]-4-(pyridin-3-yl)piperazine
1-ethyl-3-[3-(pyridin-3-yl)propyl]-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
1-[2-butyl-5-oxo-4-(3-phenylphenyl)piperazin-1-yl]butane-1,2-dione
N-{3-[2-(4-methylpentyl)morpholin-4-yl]-3-oxopropyl}acetamide