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2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-fluoro-N-methylpyrimidin-4-amine
2-(azepan-1-yl)-N-[3-(oxolan-3-yl)propyl]acetamide
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-5-oxopyrrolidine-2-carboxamide
[(2S,4R)-4-(dimethylamino)-1-[5-(3-methoxyphenyl)furan-2-carbonyl]pyrrolidin-2-yl]methanol
9-(2-methoxypyridine-4-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-cyclopropyl-1,4,6-trimethyl-N-{[4-(methylsulfanyl)phenyl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
ethyl 2-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-2-yl]acetate
N-(2-hydroxyethyl)-N-methyl-1-(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
3-(pyridin-2-yl)-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-1H-pyrazole-5-carboxamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
(3R,4S)-1-[(3,5-difluoro-4-methoxyphenyl)methyl]-3,4-dimethylpiperidin-4-ol
1-[1-(1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]piperidin-4-ol
5-[({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}(methyl)amino)methyl]-N-methylpyrimidin-2-amine
N-[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
2-{1-[5-(3-acetylphenoxymethyl)-1H-pyrazol-3-yl]-N-methylformamido}-N-methylacetamide
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-ethyl-5-methyl-1H-pyrazole-4-carboxamide
3-[5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-2,6-dimethoxypyridine
(4-{[(benzylsulfamoyl)amino]methyl}phenyl)methanol
3-(3-hydroxyphenyl)-1-{2-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}propan-1-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,6-dimethoxypyrimidine-4-carboxamide
4-(4-{1-[3-(4-methoxyphenyl)propyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
1-cyclopropyl-N-{2-[ethyl(3-methylphenyl)amino]ethyl}-1H-pyrrole-2-carboxamide
3-methyl-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}benzamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methyl-1,3-thiazole-5-carboxamide
methyl (2S,3S)-2-{[1-cyclohexyl-4-oxo-5-(pyrrolidine-1-carbonyl)-1,4-dihydropyridin-3-yl]formamido}-3-methylpentanoate
1-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}-1,4-diazepan-5-one
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}propanamide
2-{1-ethyl-8-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
4-(4-fluorophenoxy)-1-[(3-phenyloxolan-3-yl)methyl]piperidine
4-methoxy-6-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-2-amine
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}pyridazine-3-carboxamide
N-(4-acetylphenyl)-3-(2-phenylacetyl)piperidine-1-carboxamide
3-(3-fluoro-4-phenylbenzoyl)-1-(1-methylpiperidin-4-yl)piperidine
1-{4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxybenzoyl}piperazine
2-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
3-({[1-(methoxymethyl)cyclopentyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-{3-[3-(1H-indol-3-ylmethyl)-4H-1,2,4-triazol-4-yl]phenyl}ethan-1-one
N-(2,3-dihydro-1H-inden-4-yl)-4-(1,3-thiazol-2-yl)piperazine-1-carboxamide
(2S)-2-amino-N-ethyl-3-(1H-imidazol-4-yl)-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]propanamide
1-(1-benzylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
3-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}pyridin-2-amine
N-(1-hydroxybutan-2-yl)-5-methyl-N-[(2-methylphenyl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
2-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)acetamide
1-cyclopentyl-N-ethyl-5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[(4-methoxyphenyl)methyl]-4-methyl-5-[1-(pyridin-4-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
(3aR,6aR)-2-cyclopropanecarbonyl-N-[(3-methyl-1H-pyrazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-4-(3-methoxypyrazin-2-yl)piperazin-2-yl}ethan-1-ol
(4aS,7aR)-1-(2-cyclohexylethyl)-4-[2-(dimethylamino)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[3-(3-fluorophenyl)oxolan-3-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine