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1-(1-benzofuran-2-ylmethyl)-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
5-cyclopropanecarbonyl-1'-(2-ethylpyrimidine-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(methoxymethyl)-5-{[4-(piperidine-1-carbonyl)piperidin-1-yl]methyl}pyrimidine
3-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl}-4,5,6,7-tetrahydro-1,2-benzoxazole
2-[4-(4-benzylpiperazine-1-carbonyl)-5-methyl-1H-pyrazol-1-yl]-4-(2-fluorophenyl)pyrimidine
3-(2-chloro-5-sulfamoylphenyl)-1-[3-(morpholin-4-yl)propyl]urea
N-methyl-2-(morpholin-4-yl)-2-(pyridin-3-yl)-N-(thian-4-yl)acetamide
2-(2,3-difluoro-4-pentylphenyl)-N,N-dimethylpyridine-3-carboxamide
N-[2-({8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}amino)ethyl]pyridine-4-carboxamide
1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine
4-(1,3-benzothiazol-2-yl)-2-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}phenol
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-N-phenylpiperidin-3-amine
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
(4S)-1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
(1S,5R)-3-benzyl-6-(4-methoxy-3-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
2-(2-hydroxypropyl)-9-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1H-pyrrole
1-(2-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}pyrimidin-4-yl)pyrrolidin-3-ol
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-[2-(morpholin-4-ylmethyl)piperidin-1-yl]acetamide
4-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}-2,6-dimethoxyphenol
[7-(5-fluoropyrimidin-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methanamine
1-(5-{[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-methyl-1,3-oxazole-5-carboxamide
4-benzyl-3-ethyl-1-(4-propylpyrimidine-5-carbonyl)-1,4-diazepan-5-one
1-acetyl-N-[(3R,4S)-1-[(methylcarbamoyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]piperidine-4-carboxamide
(2S,4S)-4-amino-1-[2-hydroxy-6-(trifluoromethyl)pyridine-3-carbonyl]-N-methylpyrrolidine-2-carboxamide
(2R)-3-(benzyloxy)-2-({2-methylthieno[2,3-d]pyrimidin-4-yl}amino)propan-1-ol
1-{7-benzyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidine-3-carbonitrile
2-cyclohexyl-1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
3-{[2-(methoxymethyl)-1,3-benzoxazol-5-yl]methyl}-1λ6-thiane-1,1-dione
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]cycloheptanecarboxamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]-1H-pyrazole-3-carboxamide
N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-3-(thiophen-3-yl)-1H-pyrazole-5-carboxamide
3-fluoro-2-hydroxy-N-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}benzamide
2-({[(3R,4R)-1-(4,6-dimethylpyrimidin-2-yl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
(3R,4R)-N-(2-chlorophenyl)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidine-1-carboxamide
5-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-2-(methylsulfanyl)-3,4-dihydropyrimidin-4-one
2-[(2E)-3-phenylprop-2-en-1-yl]-8-(pyrazine-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(3R,4R)-4-(azepan-1-yl)-1-{[2-(cyclopentyloxy)phenyl]methyl}piperidin-3-ol
2-[1-(1-methylpiperidin-4-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]pyridine
1-(cyclohex-3-en-1-ylmethyl)-4-(2-methylphenoxy)piperidine-4-carboxylic acid
(3S,4R)-4-(2-methylphenyl)-1-[2-oxo-2-(piperidin-1-yl)ethyl]pyrrolidine-3-carboxylic acid
6-ethyl-2-methyl-N-(5-oxo-1-phenylpyrrolidin-3-yl)quinoline-4-carboxamide
N-({1-[(2E)-but-2-en-1-yl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)-2-acetamidobenzamide
2-benzyl-N-[3-(1H-1,2,4-triazol-1-yl)propyl]-1,3-thiazole-4-carboxamide
2-(2-methoxyphenyl)-5-(quinoxalin-6-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-2-methyl-N-(2-methylpropyl)pyridine-3-carboxamide
5-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-1-methyl-1H-1,2,3,4-tetrazole
2-(4-hydroxy-4-phenylpiperidin-1-yl)-2-[3-(methoxymethyl)phenyl]acetic acid
2-{4-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine